SCHEMBL365912

SCHEMBL365912

O=C(O)c1c2ccccc2n2cc(C(=O)C(F)(F)F)ccc12

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.45
HTT P42858 1/20 0.43
KDM4E B2RXH2 3/20 0.43
AGTR1 P30556 3/20 0.40
IDO1 P14902 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
EGFR P00533 2/20 0.38
RORC P51449 4/20 0.38
SRC P12931 1/20 0.37
PLA2G2D Q9UNK4 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C9 P11712 2/20 0.35
CYP3A4 P08684 1/20 0.35
MLYCD O95822 2/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365635 0.88 IDO1 (0.44) CES1HTTKDM4EIDO1HTR2A
SCHEMBL365935 0.85 KDM4E (0.47) KDM4EAGTR1EGFRRORCSRC
SCHEMBL367091 0.84 KMT2A (0.44) HTTKDM4EEGFRSRCALDH1A1
SCHEMBL366876 0.81 EGFR (0.44) KDM4EAGTR1EGFRRORCSRC
SCHEMBL366811 0.81 EGFR (0.44) KDM4EAGTR1EGFRSRCALDH1A1
SCHEMBL366000 0.80 ELANE (0.47) HTTALDH1A1
SCHEMBL365000 0.78 HTT (0.42) CES1HTTKDM4EIDO1ALDH1A1
SCHEMBL365911 0.78 CES1 (0.42) CES1HTTKDM4EAGTR1IDO1
SCHEMBL367205 0.78 EGFR (0.45) KDM4EAGTR1EGFRRORCSRC
SCHEMBL366371 0.78 EGFR (0.45) KDM4EAGTR1EGFRSRCALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed