SCHEMBL366811

SCHEMBL366811

NC(=O)c1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.44
AGTR1 P30556 4/20 0.42
KDM4E B2RXH2 2/20 0.41
SRC P12931 2/20 0.40
POLB P06746 2/20 0.40
CYP3A4 P08684 1/20 0.40
PARP1 P09874 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
FGFR1 P11362 1/20 0.40
NPC1 O15118 3/20 0.39
ELANE P08246 1/20 0.39
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367764 0.91 EGFR (0.45) EGFRKDM4ESRCPOLBCYP3A4
SCHEMBL365935 0.89 KDM4E (0.47) EGFRAGTR1KDM4ESRCPOLB
SCHEMBL365259 0.88 KDM4E (0.44) EGFRAGTR1KDM4ESRCCYP3A4
SCHEMBL366876 0.85 EGFR (0.44) EGFRAGTR1KDM4ESRCPOLB
SCHEMBL367205 0.81 EGFR (0.45) EGFRAGTR1KDM4ESRCPOLB
SCHEMBL365912 0.81 CES1 (0.45) EGFRAGTR1KDM4ESRCPOLB
SCHEMBL366371 0.81 EGFR (0.45) EGFRAGTR1KDM4ESRCPOLB
SCHEMBL367330 0.81 EGFR (0.46) EGFRKDM4ESRCPOLBNPC1
SCHEMBL366888 0.80 EGFR (0.44) EGFRAGTR1KDM4ESRCPOLB
SCHEMBL366810 0.78 PTGS2 (0.45) EGFRKDM4EPOLBCYP3A4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed