SCHEMBL366789

SCHEMBL366789

CN(C)C(=O)c1cc(O)c2c(C(=O)O)c3ccccn3c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
PTGS2 P35354 1/20 0.37
BAZ2B Q9UIF8 2/20 0.36
BAZ2A Q9UIF9 2/20 0.36
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
ERN1 O75460 2/20 0.36
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
RORC P51449 1/20 0.35
ACSS2 Q9NR19 1/20 0.35
AKR1C3 P42330 1/20 0.34
RARG P13631 1/20 0.34
ACLY P53396 1/20 0.34
PMM2 O15305 1/20 0.34
MPI P34949 1/20 0.34
PHOSPHO1 Q8TCT1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364537 0.89 BAZ2B (0.38) BAZ2BBAZ2AERN1EGFRSRC
SCHEMBL366820 0.87 IDO1 (0.43) IDO1PTGS2BAZ2BBAZ2AFNTA
SCHEMBL365788 0.86 BAZ2B (0.45) IDO1PTGS2BAZ2BBAZ2AFNTA
SCHEMBL366033 0.84 NPC1 (0.40) IDO1PTGS2FNTAFNTBERN1
SCHEMBL367255 0.83 PTGS2 (0.42) IDO1PTGS2BAZ2BBAZ2AFNTA
SCHEMBL367204 0.82 RORC (0.43) IDO1PTGS2FNTAFNTBEGFR
SCHEMBL367176 0.82 HTR6 (0.38) IDO1PTGS2ACSS2KDM4EMEN1
SCHEMBL365212 0.80 KMT2A (0.39) IDO1PTGS2BAZ2BBAZ2AKDM4E
SCHEMBL365022 0.78 PTGS2 (0.39) IDO1PTGS2BAZ2BBAZ2AFNTA
SCHEMBL367221 0.75 BAZ2B (0.42) PTGS2BAZ2BBAZ2AFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed