SCHEMBL3661420

SCHEMBL3661420

CN(C)C(=O)COc1cc(-c2ccnc(N)n2)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.44
PDPK1 O15530 2/20 0.44
AURKA O14965 2/20 0.44
CHUK O15111 1/20 0.44
RPS6KB1 P23443 1/20 0.44
KDR P35968 1/20 0.44
TGFBR1 P36897 1/20 0.44
SYK P43405 1/20 0.44
JAK3 P52333 1/20 0.44
ROCK1 Q13464 1/20 0.44
AURKB Q96GD4 1/20 0.44
MAP3K5 Q99683 1/20 0.44
KMO O15229 2/20 0.43
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPK1 P28482 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3661410 0.87 CDC7 (0.50) CDK2KMOPOLBCAMKK2ROCK2
SCHEMBL3656028 0.79 ROCK2 (0.60) CDK2PDPK1AURKACHUKRPS6KB1
SCHEMBL3723069 0.77 ROCK2 (0.65) ROCK1MEN1ALDH1A1MAPK1KMT2A
SCHEMBL2368605 0.74 ALDH1A1 (0.47) MEN1ALDH1A1MAPK1KMT2AKDM4E
SCHEMBL1987965 0.72 MEN1 (0.48) MEN1ALDH1A1MAPK1KMT2AKDM4E
SCHEMBL3656027 0.71 CDC7 (0.50) CDK2KMOCAMKK2ROCK2CDC7
SCHEMBL3044785 0.69 KMO (0.55) CDK2PDPK1AURKACHUKRPS6KB1
SCHEMBL3713494 0.69 CDK2 (0.39) CDK2PDPK1AURKACHUKRPS6KB1
SCHEMBL3720566 0.67 KMO (0.43) CDK2PDPK1AURKACHUKRPS6KB1
SCHEMBL3664825 0.67 KMO (0.57) CDK2PDPK1KMOHSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed