SCHEMBL366695

SCHEMBL366695

N#CCOc1cc(OCCc2cccnc2)c2c(C#N)c3ccccc3n2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CYP11B2 P19099 7/20 0.40
CYP11B1 P15538 6/20 0.40
CYP19A1 P11511 3/20 0.40
MAPK12 P53778 1/20 0.36
MAPK14 Q16539 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
APP P05067 1/20 0.34
SNCA P37840 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
TSHR P16473 2/20 0.34
HTT P42858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365082 0.91 CYP11B2 (0.40) CYP11B2CYP11B1KDM4EALDH1A1HPGD
SCHEMBL365103 0.90 MAPT (0.38) CYP11B2CYP11B1CYP19A1KDM4EALDH1A1
SCHEMBL364643 0.86 CYP11B1 (0.40) MKNK1MKNK2CYP11B2CYP11B1CYP19A1
SCHEMBL366016 0.85 MAPK12 (0.39) MKNK1MKNK2CYP11B2CYP11B1CYP19A1
SCHEMBL366915 0.84 PSEN1 (0.37) ALDH1A1LMNAMAPTTSHRHTT
SCHEMBL365402 0.83 PSEN1 (0.38) KDM4EALDH1A1FNTAFNTBPGGT1B
SCHEMBL366906 0.79 HTT (0.37) KDM4EALDH1A1LMNAMAPTTSHR
SCHEMBL366694 0.78 MKNK1 (0.41) MKNK1MKNK2CYP11B2CYP11B1CYP19A1
SCHEMBL367194 0.77 GPR132 (0.38) HTTCYP1A2CYP3A4CYP2C9
SCHEMBL365965 0.76 ACVR2A (0.38) KDM4EAPPSNCALMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed