SCHEMBL367194

SCHEMBL367194

N#CCOc1cc(OCc2cccnc2)c2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 10/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
MET P08581 1/20 0.37
IKBKB O14920 1/20 0.37
HTT P42858 1/20 0.37
LRRK2 Q5S007 1/20 0.36
CMKLR2 P46091 1/20 0.36
CMKLR1 Q99788 1/20 0.36
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365965 0.92 ACVR2A (0.38) GPR132CYP1A2CYP3A4CYP2C9MET
SCHEMBL364643 0.91 CYP11B1 (0.40) CYP1A2CYP3A4CYP2C9HTT
SCHEMBL365082 0.85 CYP11B2 (0.40) CYP1A2CYP3A4CYP2C9IKBKBHTR1A
SCHEMBL366016 0.84 MAPK12 (0.39) CYP1A2CYP3A4CYP2C9HTT
SCHEMBL366073 0.83 ALKBH1 (0.36)
SCHEMBL365106 0.82 KMT2A (0.39) HTT
SCHEMBL367671 0.80 PSEN1 (0.39)
SCHEMBL367193 0.79 GPR132 (0.38) GPR132METIKBKBCMKLR2CMKLR1
SCHEMBL367347 0.78 KMT2A (0.38)
SCHEMBL366565 0.77 ALDH1A1 (0.39) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed