SCHEMBL366016

SCHEMBL366016

N#CCOc1cc(OCCc2cccnc2)c2c(C(N)=O)c3ccccc3n2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK12 P53778 1/20 0.39
MAPK14 Q16539 1/20 0.39
CYP11B1 P15538 4/20 0.38
CYP11B2 P19099 4/20 0.38
CYP19A1 P11511 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
CNR2 P34972 2/20 0.36
HTT P42858 2/20 0.35
KDM4E B2RXH2 2/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
APP P05067 1/20 0.34
SNCA P37840 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364643 0.92 CYP11B1 (0.40) MAPK12MAPK14CYP11B1CYP11B2CYP19A1
SCHEMBL365965 0.92 ACVR2A (0.38) CYP1A2CYP3A4CYP2C9HTTKDM4E
SCHEMBL364641 0.90 PLK1 (0.38) CNR2SMN1; SMN2CNR1
SCHEMBL366695 0.85 MKNK1 (0.41) MAPK12MAPK14CYP11B1CYP11B2CYP19A1
SCHEMBL367249 0.85 MEN1 (0.36) HTTLMNA
SCHEMBL365786 0.85 ALDH1A1 (0.38) HTTLMNA
SCHEMBL367194 0.84 GPR132 (0.38) CYP1A2CYP3A4CYP2C9HTT
SCHEMBL366073 0.83 ALKBH1 (0.36) CNR2KDM4ESMN1; SMN2CNR1
SCHEMBL366807 0.81 MCL1 (0.33) HTTTSHRLMNASMN1; SMN2
SCHEMBL367225 0.81 KMT2A (0.40) CNR2HTTKDM4ETSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed