SCHEMBL366906

SCHEMBL366906

Cc1cnc(CCCOc2cc(OCC#N)cn3c2c(C#N)c2ccccc23)o1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 6/20 0.37
MAPT P10636 6/20 0.37
LMNA P02545 5/20 0.37
TSHR P16473 3/20 0.37
POLB P06746 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
MAPK1 P28482 4/20 0.33
L3MBTL1 Q9Y468 4/20 0.33
TDP1 Q9NUW8 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MCL1 Q07820 1/20 0.32
ALDH1A1 P00352 2/20 0.31
STAT3 P40763 1/20 0.31
MTNR1B P49286 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366831 0.86 MCL1 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL366807 0.85 MCL1 (0.33) HTTMAPTLMNATSHRPSEN1
SCHEMBL365103 0.81 MAPT (0.38) HTTMAPTLMNATSHRPOLB
SCHEMBL366905 0.80 KDM4E (0.37) HTTMAPTLMNATSHRPOLB
SCHEMBL366695 0.79 MKNK1 (0.41) HTTMAPTLMNATSHRPOLB
SCHEMBL365402 0.77 PSEN1 (0.38) HTTMAPTLMNATSHRPOLB
SCHEMBL366915 0.76 PSEN1 (0.37) HTTMAPTLMNATSHRPOLB
SCHEMBL365082 0.75 CYP11B2 (0.40) MAPTNPSR1ALDH1A1MEN1KMT2A
SCHEMBL366830 0.72 ALDH1A1 (0.35) HTTMAPTLMNAPOLBPSEN1
SCHEMBL366073 0.67 ALKBH1 (0.36) MAPTPOLBNPSR1PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed