SCHEMBL364643

SCHEMBL364643

N#CCOc1cc(OCCc2cccnc2)c2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.40
CYP11B2 P19099 7/20 0.40
CYP19A1 P11511 3/20 0.40
MAPK12 P53778 1/20 0.39
MAPK14 Q16539 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
GCK P35557 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP3A4 P08684 1/20 0.37
CNR2 P34972 1/20 0.36
HTT P42858 2/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366016 0.92 MAPK12 (0.39) CYP11B1CYP11B2CYP19A1MAPK12MAPK14
SCHEMBL367194 0.91 GPR132 (0.38) CYP1A2CYP2C9CYP3A4HTT
SCHEMBL366073 0.91 ALKBH1 (0.36) CNR2KDM4EALDH1A1
SCHEMBL366695 0.86 MKNK1 (0.41) CYP11B1CYP11B2CYP19A1MAPK12MAPK14
SCHEMBL367347 0.85 KMT2A (0.38) LMNAALDH1A1
SCHEMBL366565 0.84 ALDH1A1 (0.39) HTTALDH1A1
SCHEMBL364641 0.84 PLK1 (0.38) CNR2ALDH1A1
SCHEMBL365965 0.84 ACVR2A (0.38) CYP1A2CYP2C9CYP3A4HTTKDM4E
SCHEMBL366831 0.81 MCL1 (0.35) ALDH1A1
SCHEMBL365106 0.81 KMT2A (0.39) HTTKDM4ELMNATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed