SCHEMBL365213

SCHEMBL365213

CN(C)C(=O)Oc1cc(O)c2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NCEH1 Q6PIU2 5/20 0.38
RAB9A P51151 2/20 0.38
EGFR P00533 2/20 0.36
SRC P12931 1/20 0.36
LMNA P02545 3/20 0.36
MAOB P27338 1/20 0.35
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35
S1PR3 Q99500 1/20 0.35
MEN1 O00255 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TSPO P30536 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365256 0.90 EGFR (0.40) PKMKMT2AALDH1A1NCEH1RAB9A
SCHEMBL367616 0.89 NCEH1 (0.46) PKMKMT2AALDH1A1NCEH1RAB9A
SCHEMBL367734 0.86 ATM (0.40) PKMKMT2AALDH1A1NCEH1RAB9A
SCHEMBL366828 0.81 PKM (0.46) PKMKMT2AALDH1A1NCEH1RAB9A
SCHEMBL365189 0.80 ACHE (0.37) ALDH1A1NCEH1ACHES1PR3
SCHEMBL366116 0.80 CA1 (0.41) EGFR
SCHEMBL366790 0.80 EGFR (0.41) KMT2AALDH1A1EGFRSRCMEN1
SCHEMBL365769 0.80 LTB4R (0.39) PKMKMT2AALDH1A1LMNATSHR
SCHEMBL367671 0.78 PSEN1 (0.39) ALDH1A1EGFRTSHR
SCHEMBL365593 0.78 MRGPRX4 (0.39) PKMACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed