SCHEMBL5760090

SCHEMBL5760090

COc1cccc2c([C@@H](O)CN3CCN(CCCCc4ccccc4)CC3)ccnc12

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.47
SIGMAR1 Q99720 5/20 0.47
EBP Q15125 2/20 0.43
TMEM97 Q5BJF2 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
EBPL Q9BY08 1/20 0.42
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5754351 0.90 SIGMAR1 (0.47) SIGMAR1EBPTMEM97ADRA1DADRA1A
SCHEMBL6626086 0.87 HTR1A (0.47) KDM4EALDH1A1LMNAADRA1DADRA1A
SCHEMBL5757154 0.81 L3MBTL1 (0.54) KDM4EALDH1A1LMNAADRA1DADRA1A
SCHEMBL5757405 0.80 SLC2A1 (0.59) SIGMAR1KDM4EALDH1A1HTR1A
SCHEMBL5777034 0.80 HTR1A (0.49) KDM4EALDH1A1LMNAADRA1DADRA1A
SCHEMBL5760601 0.79 RECQL (0.45) ABCB1KDM4EALDH1A1LMNAADRA1D
SCHEMBL5776914 0.76 MEN1 (0.40) TMEM97KDM4EALDH1A1LMNAADRA1D
SCHEMBL5754921 0.75 MAPK1 (0.43) ABCB1KDM4EALDH1A1LMNAADRA1D
SCHEMBL5773715 0.75 SLC2A1 (0.39) TMEM97KDM4EALDH1A1ADRA1BDRD2
SCHEMBL6977618 0.75 HTR4 (0.46) TMEM97KDM4EALDH1A1ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343765-B1 QUINOLINES AND NITROGENATED DERIVATIVES THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERAZINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2006-11-22 EP claimed