SCHEMBL370651

SCHEMBL370651

CC(=O)C(c1ccc(C)cc1)(c1ccc(Br)cc1)c1cc(Cl)ncc1F

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.32
RAB9A P51151 4/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 2/20 0.32
ALDH1A1 P00352 3/20 0.32
HTT P42858 2/20 0.32
KCNQ3 O43525 4/20 0.31
KCNQ2 O43526 4/20 0.31
KCNE1 P15382 4/20 0.31
KCNQ1 P51787 4/20 0.31
TP53 P04637 1/20 0.31
LMNA P02545 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
S1PR3 Q99500 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL371335 0.81 RAB9A (0.32) RAB9ASMN1; SMN2NPC1ALDH1A1HTT
SCHEMBL370104 0.78 RAB9A (0.33) HDAC1RAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL364975 0.76 GPBAR1 (0.30) GPBAR1
SCHEMBL363181 0.70 HDAC3 (0.38) HDAC1ALDH1A1HDAC3HDAC2HDAC6
SCHEMBL362323 0.70 KCNN4 (0.41) HDAC1ALDH1A1KCNE1KCNQ1MEN1
SCHEMBL363897 0.68 AR (0.36) RAB9ASMN1; SMN2NPC1ALDH1A1MEN1
SCHEMBL362974 0.68 KCNN4 (0.35) RAB9AALDH1A1KCNE1KCNQ1HDAC6
SCHEMBL361971 0.65 NR1H2 (0.37) RAB9ASMN1; SMN2NPC1ALDH1A1HTT
SCHEMBL364587 0.65 SORT1 (0.34) ALDH1A1
SCHEMBL363084 0.65 SORT1 (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed