SCHEMBL371748

SCHEMBL371748

c1ccc(Cc2ccsc2Cc2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.46
BCL2 P10415 1/20 0.43
BCL2L1 Q07817 1/20 0.43
LTB4R Q15722 6/20 0.41
HTR2A P28223 1/20 0.41
ALOX5 P09917 1/20 0.38
PTPN1 P18031 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5109182 0.86 TSHR (0.43) CALM1BCL2BCL2L1LTB4RPTPN1
SCHEMBL5117305 0.86 BCL2 (0.44) CALM1BCL2BCL2L1LTB4RHTR2A
SCHEMBL10718336 0.81 LTB4R (0.49) BCL2BCL2L1LTB4RKMT2AALOX15
SCHEMBL10720297 0.81 LTB4R (0.49) LTB4RPTPN1MEN1KMT2AALOX15
SCHEMBL29480061 0.80 KEAP1 (0.53) BCL2BCL2L1HTR2AALOX5PTPN1
SCHEMBL7585710 0.78 MET (0.35) BCL2BCL2L1LTB4RMEN1KMT2A
SCHEMBL9024878 0.77 CALM1 (0.44) CALM1BCL2BCL2L1LTB4RHTR2A
SCHEMBL10947990 0.77 CALM1 (0.44) CALM1BCL2BCL2L1HTR2AALOX5
SCHEMBL6947065 0.77 ADRA1D (0.46) CALM1ALOX5PTPN1MEN1KMT2A
SCHEMBL16612937 0.77 CALM1 (0.44) CALM1BCL2BCL2L1HTR2AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 136 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1757645-A Material contg. thiophene spirane structure, its synthesis and application UNIV FUDAN (CN) 2006-04-12 CN claimed
US-6809229-B2 USED EITHER AS CATALYST AND/OR CATALYST SUPPORTS IN FLUID PHASE CATALYTIC CHEMICAL REACTIONS, SUCH AS HYDROGENATION, HYDRODESULFURIZATION, OXIDATION AND ISOMERIZATION HYPERION CATALYSIS INTERNATIONAL, INC. 2004-10-26 US claimed
US-20020121460-A1 Method of using carbide and/or oxycarbide containing compositions HYPERION CATALYSIS INTERNATIONAL 2002-09-05 US claimed
US-5668168-A FUNGICIDES SHAMAN PHARMACEUTICALS, INC. (US) 1997-09-16 US claimed
US-5556875-A FUNGICIDES SHAMAN PHARMACEUTICALS, INC. (US) 1996-09-17 US claimed
EP-0714297-A4 1996-07-10 EP claimed
EP-0714297-A1 NOVEL 1,2-DITHIIN ANTIINFECTIVE AGENTS SHAMAN PHARMACEUTICALS, INC. (US) 1996-06-05 EP claimed
WO-1995005817-A1 NOVEL 1,2-DITHIIN ANTIINFECTIVE AGENTS SHAMAN PHARMACEUTICALS, INC. (US) 1995-03-02 WO claimed
EP-0136469-B1 HYDROFINING PROCESS FOR HYDROCARBON-CONTAINING FEED STREAMS PHILLIPS PETROLEUM COMPANY (US) 1991-10-23 EP claimed
EP-0133649-B1 IMPROVING THE LIFE OF A CATALYST USED TO PROCESS HYDROCARBON CONTAINING FEED STREAMS PHILLIPS PETROLEUM COMPANY (US) 1988-05-11 EP claimed
US-4564441-A Hydrofining process for hydrocarbon-containing feed streams PHILLIPS PETROLEUM COMPANY (US) 1986-01-14 US claimed
EP-0136469-A1 Hydrofining process for hydrocarbon-containing feed streams PHILLIPS PETROLEUM COMPANY (US) 1985-04-10 EP claimed
EP-0133649-A1 Improving the life of a catalyst used to process hydrocarbon containing feed streams PHILLIPS PETROLEUM COMPANY (US) 1985-03-06 EP claimed
EP-2892646-B1 HYDROCONVERSION MULTI-METALLIC CATALYST CHEVRON USA INC (US) 2021-10-20 EP disclosed
EP-2791293-B1 PREPARATION OF A POST-TREATED MOLYBDENUM AMIDE ADDITIVE COMPOSITION AND LUBRICATING OIL COMPOSITIONS CONTAINING SAME CHEVRON ORONITE CO (US) 2018-09-26 EP disclosed
EP-2271652-B1 PREPARATION OF A MOLYBDENUM AMIDE ADDITIVE COMPOSITION AND LUBRICATING OIL COMPOSITIONS CONTAINING SAME CHEVRON ORONITE CO (US) 2018-04-25 EP disclosed
US-4492626-A PLATINUM WITH OXIDE PROMOTER PHILLIPS PETROLEUM COMPANY (US) 1985-01-08 US disclosed
US-4457836-A FROM PETROLEUM DISTILLATES EXXON RESEARCH AND ENGINEERING COMPANY (US) 1984-07-03 US disclosed
US-4431747-A HYDROREFINING CATALYSTS; METHANATION; HYDROTREATMENT; IMPREGNATING WITH A ORGANIC AMINE METAL COMPLEX EXXON RESEARCH AND ENGINEERING CO. (US) 1984-02-14 US disclosed
US-4430442-A HYDROREFINING CATALYSTS; CATALYST SELECTIVETY; HYDRODENITROGENIZATION EXXON RESEARCH AND ENGINEERING CO. (US) 1984-02-07 US disclosed