SCHEMBL3742268

SCHEMBL3742268

COc1cc2oc3cc(O)c(OC)c(CC=C(C)C)c3c(=O)c2c(O)c1CC=C(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 7/20 1.00
GAA P10253 7/20 1.00
SI P14410 7/20 1.00
MGAM2 Q2M2H8 7/20 1.00
IDH1 O75874 4/20 1.00
FASN P49327 4/20 1.00
RELA Q04206 3/20 1.00
SIRT2 Q8IXJ6 3/20 1.00
NFKB1 P19838 1/20 1.00
PTPN1 P18031 4/20 0.85
SMPD1 P17405 3/20 0.85
CYP19A1 P11511 3/20 0.85
NUDT1 P36639 3/20 0.85
PGAM1 P18669 3/20 0.85
AKR1B1 P15121 2/20 0.85
PDE4D Q08499 2/20 0.85
KDM4E B2RXH2 1/20 0.85
MEN1 O00255 1/20 0.85
KDM1A O60341 1/20 0.85
USP2 O75604 1/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29929598 1.00 MGAM (1.00) MGAMGAASIMGAM2IDH1
SCHEMBL29974819 1.00 MGAM (1.00) MGAMGAASIMGAM2IDH1
SCHEMBL29929664 0.93 MGAM (0.87) MGAMGAASIMGAM2IDH1
SCHEMBL3740906 0.93 MGAM (0.87) MGAMGAASIMGAM2IDH1
Mangostin SCHEMBL354735 0.92 MGAM (1.00) MGAMGAASIMGAM2IDH1
Mangostin SCHEMBL29466055 0.92 MGAM (1.00) MGAMGAASIMGAM2IDH1
Mangostin SCHEMBL29433195 0.92 MGAM (1.00) MGAMGAASIMGAM2IDH1
SCHEMBL3750432 0.91 MGAM (0.85) MGAMGAASIMGAM2IDH1
SCHEMBL30830372 0.91 MGAM (0.85) MGAMGAASIMGAM2IDH1
Mangostin SCHEMBL676010 0.91 MGAM (0.98) MGAMGAASIMGAM2IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260048096-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE RETINAL OUTER NUCLEAR LAYER (ONL), PHOTORECEPTORS, AND RETINAL THICKNESS STEALTH BIOTHERAPEUTICS INC. (US) 2026-02-19 US claimed
US-20250090621-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC. (US) 2025-03-20 US claimed
US-20250057805-A1 METHODS FOR ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF BEVEMIPRETIDE STEALTH BIOTHERAPEUTICS INC. (US) 2025-02-20 US claimed
US-20240299486-A1 ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF ELAMIPRETIDE STEALTH BIOTHERAPEUTICS INC. (US) 2024-09-12 US claimed
WO-2023230322-A1 ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF ELAMIPRETIDE STEALTH BIOTHERAPEUTICS INC. (US) 2023-11-30 WO claimed
WO-2021042001-A1 COMPOSITIONS AND METHODS RELATED TO DISSOLVED OXIDES Natural Extraction Systems, LLC (US) 2021-03-04 WO claimed
US-8461360-B2 Process for producing γ -mangostin LAILA NUTRACEUTICALS (US) 2013-06-11 US claimed
US-20100292490-A1 A PROCESS FOR PRODUCING GAMMA MANGOSTIN LAILA NUTRACEUTICALS (IN) 2010-11-18 US claimed
WO-2009093259-A2 A PROCESS FOR PRODUCING γ-MANGOSTIN GOKARAJU GANGA RAJU (IN) 2009-07-30 WO claimed
US-20260048096-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE RETINAL OUTER NUCLEAR LAYER (ONL), PHOTORECEPTORS, AND RETINAL THICKNESS STEALTH BIOTHERAPEUTICS INC. (US) 2026-02-19 US disclosed
US-20250302909-A1 METHODS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC. (US) 2025-10-02 US disclosed
US-20250090621-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC. (US) 2025-03-20 US disclosed
US-20250057805-A1 METHODS FOR ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF BEVEMIPRETIDE STEALTH BIOTHERAPEUTICS INC. (US) 2025-02-20 US disclosed
US-20240299486-A1 ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF ELAMIPRETIDE STEALTH BIOTHERAPEUTICS INC. (US) 2024-09-12 US disclosed
US-20100093843-A1 NOVEL NUTRACEUTICAL AND PHARMACEUTICAL COMPOSITIONS AND USE THEREOF FOR THE TREATMENT, CO-TREATMENT OR PREVENTION OF CARTILAGE DEGRADATION OR CARTILAGE DAMAGE IN JOINTS DSM IP ASSETS B.V. (NL) 2010-04-15 US disclosed
US-20090221693-A1 NOVEL USE OF ORGANIC COMPOUNDS DSM IP ASSETS B.V. (NL) 2009-09-03 US disclosed
US-20090221693-A1 NOVEL USE OF ORGANIC COMPOUNDS DSM IP ASSETS B.V. (NL) 2009-09-03 US disclosed
WO-2009093259-A2 A PROCESS FOR PRODUCING γ-MANGOSTIN GOKARAJU GANGA RAJU (IN) 2009-07-30 WO disclosed
WO-2008031572-A1 NOVEL NUTRACEUTICAL AND PHARMACEUTICAL COMPOSITIONS AND USE THEREOF FOR THE TREATMENT, CO-TREATMENT OR PREVENTION OF CARTILAGE DEGRADATION OR CARTILAGE DAMAGE IN JOINTS DSM IP ASSETS B.V. (NL) 2008-03-20 WO disclosed
WO-2007128465-A1 XANTHONE DERIVATIVE FOR THE TREATMENT OF MUSCULAR DISORDERS DSM IP ASSETS B.V. (NL) 2007-11-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260048096-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE RETINAL OUTER NUCLEAR LAYER (ONL), PHOTORECEPTORS, AND RETINAL THICKNESS NR2E3, ALDH1A2, PDE6D MGAM 4027/4885GAA 2896/4885SI 290/4885
US-20250090621-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION PDE6C, PDE6A, PDE6B MGAM 1971/4885GAA 2047/4885SI 1825/4885
US-20250302909-A1 METHODS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION PDE6C, PDE6A, PDE6B MGAM 1422/4885GAA 1324/4885SI 1356/4885
US-20100292490-A1 A PROCESS FOR PRODUCING GAMMA MANGOSTIN SOST, CYP51A1, GNMT MGAM 39/4885GAA 342/4885SI 201/4885
US-20250057805-A1 METHODS FOR ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF BEVEMIPRETIDE MRGPRX2, MRGPRX4, MRGPRX1 MGAM 136/4885GAA 891/4885SI 119/4885
US-20100093843-A1 NOVEL NUTRACEUTICAL AND PHARMACEUTICAL COMPOSITIONS AND USE THEREOF FOR THE TREATMENT, CO-TREATMENT OR PREVENTION OF CARTILAGE DEGRADATION OR CARTILAGE DAMAGE IN JOINTS COL2A1, COL1A1, COL14A1 MGAM 2749/4885GAA 1332/4885SI 847/4885
US-20090221693-A1 NOVEL USE OF ORGANIC COMPOUNDS CPT1B, MTPN, SOST MGAM 1028/4885GAA 176/4885SI 552/4885
US-20240299486-A1 ADDRESSING INJECTION SITE REACTIONS ASSOCIATED WITH THE ADMINISTRATION OF ELAMIPRETIDE MRGPRX2, MRGPRX1, MRGPRX4 MGAM 426/4885GAA 1690/4885SI 62/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.