SCHEMBL3782999

SCHEMBL3782999

COc1nc(NC(C)C)nc2nnc(-c3ccc(F)cc3)nc12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 5/20 0.41
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
NTRK1 P04629 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
DYRK1A Q13627 1/20 0.33
FPR2 P25090 2/20 0.31
SCN9A Q15858 2/20 0.31
MAPK14 Q16539 3/20 0.31
MAPK10 P53779 1/20 0.31
PIM1 P11309 1/20 0.31
PIM2 Q9P1W9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3787051 0.87 MEN1 (0.39) KCNH3MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL3781206 0.83 CNR2 (0.36) MEN1KMT2ASMN1; SMN2LMNANPC1
SCHEMBL3788039 0.82 MAPT (0.44) KCNH3MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL3706380 0.79 KCNH3 (0.42) KCNH3SCN9A
SCHEMBL3785711 0.79 KCNH3 (0.43) KCNH3MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL3780588 0.78 LMNA (0.42) KCNH3MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL3785163 0.73 KCNH3 (0.40) KCNH3MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL3776179 0.72 MPO (0.39) MEN1KMT2ASMN1; SMN2LMNANPC1
SCHEMBL3779747 0.71 MPO (0.38) MEN1KMT2ASMN1; SMN2LMNANPC1
SCHEMBL3787119 0.71 KCNH3 (0.39) KCNH3MEN1KMT2ALMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed