SCHEMBL3783192

SCHEMBL3783192

O=C(O)CN1CCN(CC(=O)O)CCN(CC(Cc2ccc([N+](=O)O)cc2)N(CC(=O)O)CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.34
S1PR1 P21453 1/20 0.33
OPRK1 P41145 1/20 0.32
HTR1A P08908 1/20 0.31
KCNJ1 P48048 2/20 0.31
KCNH2 Q12809 2/20 0.31
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 1/20 0.31
NR2F2 P24468 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
POLB P06746 1/20 0.31
ALDH1A1 P00352 3/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13014163 0.90 OPRK1 (0.42) OPRK1KCNJ1KCNH2KDM4ENPC1
SCHEMBL463667 0.90 OPRK1 (0.42) OPRK1KCNJ1KCNH2KDM4ENPC1
SCHEMBL408756 0.85 KCNJ1 (0.43) OPRK1KCNJ1KCNH2KDM4ENPC1
SCHEMBL13013959 0.84 LMNA (0.41) SLC6A9S1PR1RAB9ASMN1; SMN2POLB
SCHEMBL3769677 0.84 OPRK1 (0.38) SLC6A9S1PR1OPRK1HTR1AALDH1A1
SCHEMBL18021169 0.82 SIGMAR1 (0.41) OPRK1KCNJ1KCNH2
SCHEMBL22821445 0.81 S1PR1 (0.36) SLC6A9S1PR1HTR1ANPC1RAB9A
SCHEMBL18371468 0.81 ALPL (0.39) KDM4EPOLB
SCHEMBL3782596 0.80 NR1D1 (0.35) OPRK1HTR1ANPC1RAB9A
SCHEMBL18021181 0.80 SIGMAR1 (0.41) OPRK1KCNJ1KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10556873-B2 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2020-02-11 US disclosed
US-10189803-B2 Synthesis of therapeutic and diagnostic drugs centered on regioselective and stereoselective ring opening of aziridinium ions ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2019-01-29 US disclosed
US-20170008863-A1 SYNTHESIS OF THERAPEUTIC AND DIAGNOSTIC DRUGS CENTERED ON REGIOSELECTIVE AND STEREOSELECTIVE RING OPENING OF AZIRIDINIUM IONS CHONG, HYUN-SOON, PHD 2017-01-12 US disclosed
US-20160052894-A1 BIMODAL LIGANDS WITH MACROCYCLIC AND ACYCLIC BINDING MOIETIES, COMPLEXES AND COMPOSITIONS THEREOF, AND METHODS OF USING CHONG, HYUN-SOON, PHD 2016-02-25 US disclosed
US-9115094-B2 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using THE UNITED STATES OF AMERICA, NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS) (US) 2015-08-25 US disclosed
US-20100322855-A1 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2010-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10556873-B2 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using UACA, CLTC, CLTA SLC6A9 2253/4885S1PR1 3261/4885OPRK1 1962/4885
US-20160052894-A1 BIMODAL LIGANDS WITH MACROCYCLIC AND ACYCLIC BINDING MOIETIES, COMPLEXES AND COMPOSITIONS THEREOF, AND METHODS OF USING UACA, CLTC, CLTA SLC6A9 2253/4885S1PR1 3261/4885OPRK1 1962/4885
US-20170008863-A1 SYNTHESIS OF THERAPEUTIC AND DIAGNOSTIC DRUGS CENTERED ON REGIOSELECTIVE AND STEREOSELECTIVE RING OPENING OF AZIRIDINIUM IONS AZI2, ABL1, DHPS SLC6A9 822/4885S1PR1 2342/4885OPRK1 901/4885
US-10189803-B2 Synthesis of therapeutic and diagnostic drugs centered on regioselective and stereoselective ring opening of aziridinium ions AZI2, ABL1, DHPS SLC6A9 822/4885S1PR1 2342/4885OPRK1 901/4885
US-20100322855-A1 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using UACA, CLTC, PKD1 SLC6A9 2341/4885S1PR1 2492/4885OPRK1 1560/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.