SCHEMBL380132

SCHEMBL380132

C[Si](C)(C)[O-].[Na+]

nearest known ligand 0.00

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1577494 0.86 ALDH1A1 (0.30)
SCHEMBL1577864 0.86 ALDH1A1 (0.30)
SCHEMBL9618786 0.86
SCHEMBL9118174 0.86 ALDH1A1 (0.30)
SCHEMBL1577957 0.86 ALDH1A1 (0.30)
SCHEMBL25338226 0.86
Lithium Ion SCHEMBL380890 0.86
Potassium Ion SCHEMBL56363 0.86
SCHEMBL21357941 0.86
SCHEMBL5445634 0.86 ALDH1A1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 893 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026090336-A1 PROCESSES FOR PREPARING KRAS INHIBITORS INCYTE CORPORATION (US) 2026-04-30 WO claimed
EP-4720050-A1 PROCESS OF PREPARING HIV CAPSID INHIBITOR GILEAD SCIENCES, INC. (US) 2026-04-08 EP claimed
EP-4683926-A1 MONO-SUBSTITUTED TIN COMPOUNDS AND RELATED METHODS Entegris, Inc. (US) 2026-01-28 EP claimed
US-20250372660-A1 HIGH-ENERGY LITHIUM METAL BATTERIES ACHIEVED BY INORGANIC AND ORGANIC COATINGS BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) 2025-12-04 US claimed
WO-2025080589-A1 PROCESSES FOR PREPARING KRAS INHIBITORS INCYTE CORPORATION (US) 2025-04-17 WO claimed
WO-2025042679-A1 FASTER AUTOMATED ITERATIVE C-C BOND FORMATION THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2025-02-27 WO claimed
WO-2024249672-A1 PROCESS OF PREPARING HIV CAPSID INHIBITOR GILEAD SCIENCES, INC. (US) 2024-12-05 WO claimed
WO-2024227071-A1 SYNTHESIS OF DURLOBACTAM ENTASIS THERAPEUTICS LIMITED (GB) 2024-10-31 WO claimed
US-20240317781-A1 MONO-SUBSTITUTED TIN COMPOUNDS AND RELATED METHODS ENTEGRIS, INC. 2024-09-26 US claimed
WO-2024197115-A1 MONO-SUBSTITUTED TIN COMPOUNDS AND RELATED METHODS ENTEGRIS, INC. (US) 2024-09-26 WO claimed
EP-0575463-A1 C-TERMINAL PEPTIDE SEQUENCING USING DIPHENYL PHOSPHOROISOTHIOCYANATIDATE AND PYRIDINE CITY OF HOPE (US) 1993-12-29 EP claimed
WO-1993011436-A1 C-TERMINAL PEPTIDE SEQUENCING USING DIPHENYL PHOSPHOROISOTHIOCYANATIDATE AND PYRIDINE CITY OF HOPE (US) 1993-06-10 WO claimed
US-5180807-A C-terminal peptide or protein sequencing reagent and method CITY OF HOPE (US) 1993-01-19 US claimed
EP-0483162-A4 SEQUENTIAL C-TERMINAL DEGRADATION OF PEPTIDES AND PROTEINS 1993-01-07 EP claimed
EP-0483162-A1 SEQUENTIAL C-TERMINAL DEGRADATION OF PEPTIDES AND PROTEINS. HOPE CITY (US) 1992-05-06 EP claimed
WO-1991018008-A1 SEQUENTIAL C-TERMINAL DEGRADATION OF PEPTIDES AND PROTEINS CITY OF HOPE (US) 1991-11-28 WO claimed
US-5059540-A Coupling the peptide with a silane isothiocyanate to form a thiohydantoin derivative CITY OF HOPE (US) 1991-10-22 US claimed
EP-0200307-B1 IMPROVED PROCESS FOR PRODUCTION OF QUINOLINE-3-CARBOXYLIC ACID ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1989-12-20 EP claimed
EP-0200307-A1 Improved process for production of quinoline-3-carboxylic acid antibacterial agents WARNER-LAMBERT COMPANY (US) 1986-11-05 EP claimed
US-4003917-A Siloxanediolate complexes and preparation thereof GENERAL ELECTRIC COMPANY (US) 1977-01-18 US claimed