SCHEMBL3828535

SCHEMBL3828535

CC(CC(=O)N(Cc1ccc(N2CCN(C)CC2)nc1)c1ccc(F)cc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 1/20 0.45
TSHR P16473 1/20 0.45
EP300 Q09472 1/20 0.45
RORC P51449 1/20 0.42
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
HTR1A P08908 2/20 0.39
DRD4 P21917 2/20 0.39
HTR2A P28223 2/20 0.39
SLC6A4 P31645 2/20 0.39
DRD3 P35462 2/20 0.39
POLB P06746 1/20 0.39
MAPK14 Q16539 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ME2 P23368 1/20 0.38
ME1 P48163 1/20 0.38
ME3 Q16798 1/20 0.38
CCR5 P51681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3829302 0.85 ALDH1A1 (0.50) ALDH1A1KDM4ETSHREP300RORC
SCHEMBL3830332 0.83 MEN1 (0.45) ALDH1A1KDM4ETSHREP300RORC
SCHEMBL8184147 0.81 L3MBTL1 (0.47) ALDH1A1KDM4ETSHRHTR1ADRD4
SCHEMBL3823632 0.80 L3MBTL1 (0.45) ALDH1A1KDM4ETSHREP300RORC
SCHEMBL3826601 0.80 RAB9A (0.48) ALDH1A1KDM4ETSHRHTR1ADRD4
SCHEMBL8184144 0.79 L3MBTL1 (0.44) ALDH1A1KDM4ETSHREP300RORC
SCHEMBL8177578 0.79 OPRM1 (0.45) ALDH1A1KDM4ETSHREP300CHRM5
SCHEMBL3053852 0.79 ME2 (0.43) ALDH1A1KDM4ETSHREP300CHRM5
SCHEMBL3827091 0.79 L3MBTL1 (0.44) ALDH1A1KDM4ETSHREP300CHRM5
SCHEMBL3860025 0.79 L3MBTL1 (0.53) ALDH1A1KDM4ETSHREP300CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097379-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-09-09 EP claimed
WO-2008073936-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed