SCHEMBL3829302

SCHEMBL3829302

CN1CCN(c2ccc(CN(C(=O)CCc3ccccc3)c3ccc(F)cc3)cn2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
TSHR P16473 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ME2 P23368 2/20 0.49
ME1 P48163 2/20 0.49
ME3 Q16798 2/20 0.49
CHRM5 P08912 2/20 0.48
CHRM1 P11229 2/20 0.48
CHRM3 P20309 2/20 0.48
HTR1A P08908 3/20 0.46
DRD4 P21917 3/20 0.46
HTR2A P28223 3/20 0.46
DRD3 P35462 3/20 0.46
SLC6A4 P31645 2/20 0.46
EP300 Q09472 1/20 0.46
MLYCD O95822 1/20 0.44
DRD2 P14416 2/20 0.43
HTR2C P28335 2/20 0.43
HTR7 P34969 2/20 0.43
DRD1 P21728 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3830332 0.86 MEN1 (0.45) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL3828535 0.85 ALDH1A1 (0.45) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL8184147 0.83 L3MBTL1 (0.47) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL3826601 0.83 RAB9A (0.48) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL3823632 0.83 L3MBTL1 (0.45) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL3053852 0.82 ME2 (0.43) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL8177578 0.82 OPRM1 (0.45) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL4737954 0.82 KDM4E (0.45) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL3827091 0.82 L3MBTL1 (0.44) ALDH1A1TSHRKDM4EME2ME1
SCHEMBL3860025 0.82 L3MBTL1 (0.53) ALDH1A1TSHRKDM4EME2ME1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097379-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-09-09 EP claimed
WO-2008073936-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed
WO-2008073936-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed