SCHEMBL383482

SCHEMBL383482

CC(=O)CCC(=O)Oc1ccc([C](c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.57
ELANE P08246 5/20 0.55
ALDH1A1 P00352 3/20 0.51
HTT P42858 3/20 0.51
MAPT P10636 2/20 0.51
LMNA P02545 1/20 0.51
HSD17B10 Q99714 1/20 0.51
ESR1 P03372 4/20 0.46
MEN1 O00255 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
RECQL P46063 1/20 0.44
HIF1A Q16665 1/20 0.44
POLB P06746 1/20 0.43
SIRT5 Q9NXA8 1/20 0.43
PARP10 Q53GL7 1/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL522154 0.93 KMT2A (0.58) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL5711151 0.86 ALDH1A1 (0.57) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL22666944 0.81 ELANE (0.74) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL23843934 0.78 KMT2A (0.60) KMT2AALDH1A1HTTMAPTLMNA
SCHEMBL28340805 0.78 KMT2A (0.66) KMT2AALDH1A1HTTMAPTLMNA
SCHEMBL43742 0.76 KMT2A (0.61) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL28370277 0.76 KMT2A (0.58) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL14276948 0.76 PRSS1 (0.54) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL29947443 0.76 ALDH1A1 (0.46) KMT2AELANEALDH1A1HTTMAPT
SCHEMBL18333384 0.75 KMT2A (0.57) KMT2AALDH1A1HTTMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 110 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121719-A2 2-5A DERIVATIVES AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI-PARASITIC AGENTS Alios Biopharma, Inc. (US) 2009-11-25 EP claimed
WO-2009086192-A1 BIODEGRADABLE PHOSPHATE PROTECTED NUCLEOTIDE DERIVATIVES AND THEIR USE AS CANCER, ANTI VIRAL AND ANTI PARASITIC AGENTS ALIOS BIOPHARMA, INC. (US) 2009-07-09 WO claimed
WO-2009086201-A1 2-5A ANALOGS AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI- PARAS ITI C AGENTS ALIOS BIOPHARMA, INC. (US) 2009-07-09 WO claimed
WO-2008095040-A2 2-5A DERIVATIVES AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI-PARASITIC AGENTS ALIOS BIOPHARMA, INC. (US) 2008-08-07 WO claimed
WO-2000004062-A1 RECOVERY OF TRIARYLMETHYL HALIDE PROTECTING GROUPS CLEAVED DURING OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2000-01-27 WO claimed
EP-3160475-B1 SUBSTITUTED NUCLEOSIDES AND NUCLEOTIDES TO TREAT FILOVIRIDAE INFECTIONS JANSSEN PHARMACEUTICALS INC (US) 2024-01-03 EP disclosed
EP-3013340-B9 SUBSTITUTED NUCLEOSIDES, NUCLEOTIDES AND ANALOGS THEREOF JANSSEN PHARMACEUTICALS INC (US) 2023-10-04 EP disclosed
EP-3013340-B1 SUBSTITUTED NUCLEOSIDES, NUCLEOTIDES AND ANALOGS THEREOF JANSSEN BIOPHARMA INC (US) 2023-06-07 EP disclosed
US-20230167151-A1 SUBSTITUTED NUCLEOSIDES, NUCLEOTIDES AND ANALOGS THEREOF JANSSEN PHARMACEUTICA NV (BE) 2023-06-01 US disclosed
US-11590155-B2 Substituted nucleosides, nucleotides and analogs thereof JANSSEN PHARMACEUTICA NV (BE) 2023-02-28 US disclosed
US-11485753-B2 Substituted nucleosides, nucleotides and analogs thereof JANSSEN PHARMACEUTICA NV (BE) 2022-11-01 US disclosed
EP-3912984-A1 4'-FLUORO-NUCLEOSIDES, 4'-FLUORO-NUCLEOTIDES AND ANALOGS THEREOF FOR THE TREATMENT OF HCV Janssen BioPharma, Inc. (US) 2021-11-24 EP disclosed
US-20100240604-A1 PROTECTED NUCLEOTIDE ANALOGS ALIOS BIOPHARMA, INC. (US) 2010-09-23 US disclosed
EP-2121719-A2 2-5A DERIVATIVES AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI-PARASITIC AGENTS Alios Biopharma, Inc. (US) 2009-11-25 EP disclosed
US-20090181921-A1 2-5A ANALOGS AND THEIR METHODS OF USE ALIOS BIOPHARMA INC. (US) 2009-07-16 US disclosed
WO-2009086192-A1 BIODEGRADABLE PHOSPHATE PROTECTED NUCLEOTIDE DERIVATIVES AND THEIR USE AS CANCER, ANTI VIRAL AND ANTI PARASITIC AGENTS ALIOS BIOPHARMA, INC. (US) 2009-07-09 WO disclosed
WO-2009086201-A1 2-5A ANALOGS AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI- PARAS ITI C AGENTS ALIOS BIOPHARMA, INC. (US) 2009-07-09 WO disclosed
US-20090176732-A1 PROTECTED NUCLEOTIDE ANALOGS ALIOS BIOPHARMA INC. (US) 2009-07-09 US disclosed
US-20080207554-A1 2-5A Analogs and their Methods of Use ALIOS BIOPHARMA, INC. (US) 2008-08-28 US disclosed
WO-2008095040-A2 2-5A DERIVATIVES AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI-PARASITIC AGENTS ALIOS BIOPHARMA, INC. (US) 2008-08-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11485753-B2 Substituted nucleosides, nucleotides and analogs thereof PNP, NUDT1, NT5C2 KMT2A 3429/4885ELANE 931/4885ALDH1A1 1431/4885
US-20090176732-A1 PROTECTED NUCLEOTIDE ANALOGS NTPCR, NT5C2, PNP KMT2A 2834/4885ELANE 390/4885ALDH1A1 941/4885
US-20230167151-A1 SUBSTITUTED NUCLEOSIDES, NUCLEOTIDES AND ANALOGS THEREOF PNP, NUDT1, NT5C2 KMT2A 3429/4885ELANE 931/4885ALDH1A1 1431/4885
US-20090181921-A1 2-5A ANALOGS AND THEIR METHODS OF USE RNASEL, RNASE1, RNASEH1 KMT2A 1495/4885ELANE 447/4885ALDH1A1 1161/4885
US-20100240604-A1 PROTECTED NUCLEOTIDE ANALOGS PNP, NTPCR, TYMP KMT2A 3154/4885ELANE 1296/4885ALDH1A1 3343/4885
US-11590155-B2 Substituted nucleosides, nucleotides and analogs thereof PNP, NUDT1, NT5C3B KMT2A 3185/4885ELANE 683/4885ALDH1A1 2125/4885
US-20080207554-A1 2-5A Analogs and their Methods of Use RNASEL, RNASE1, RNASEH1 KMT2A 1855/4885ELANE 540/4885ALDH1A1 622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.