SCHEMBL396957

SCHEMBL396957

CCN1C(=O)C(=O)c2cc(C)ccc21

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARK7 Q99497 1/20 0.68
ALDH1A1 P00352 8/20 0.64
ACHE P22303 2/20 0.61
MAPT P10636 8/20 0.60
KMT2A Q03164 5/20 0.60
MEN1 O00255 4/20 0.60
LMNA P02545 4/20 0.60
POLB P06746 3/20 0.60
RCE1 Q9Y256 2/20 0.60
TDP1 Q9NUW8 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
HSP90AA1 P07900 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
TP53 P04637 2/20 0.55
KDM4E B2RXH2 1/20 0.53
AGTR1 P30556 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29862307 1.00 PARK7 (0.68) PARK7ALDH1A1ACHEMAPTKMT2A
SCHEMBL13546141 0.86 ALDH1A1 (0.65) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL7293785 0.84 ACHE (0.60) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL4625552 0.84 ALDH1A1 (0.62) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL28205978 0.83 ALDH1A1 (0.68) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL20248917 0.83 ALDH1A1 (0.50) PARK7ALDH1A1ACHEMAPTKMT2A
SCHEMBL16329852 0.81 ACHE (0.83) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL4624784 0.81 ALDH1A1 (0.63) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL16048726 0.81 ALDH1A1 (0.60) ALDH1A1ACHEMAPTKMT2AMEN1
SCHEMBL3020410 0.81 CES1 (0.67) ALDH1A1ACHEMAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250236590-A1 A METHOD FOR THE PREPARATION OF INDOLE-3-CARBOXYLIC ACID DERIVATIVES DEB INDUBHUSAN 2025-07-24 US disclosed
US-11858915-B2 Polo like kinase 4 inhibitors ORIC PHARMACEUTICALS, INC. (US) 2024-01-02 US disclosed
WO-2023067628-A1 A METHOD FOR THE PREPARATION OF INDOLE-3-CARBOXYLIC ACID DERIVATIVES COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH AN INDIAN REGISTERED BODY INCORPORATED UNDER THE REGN. OF SOC. ACT (ACT XXI OF 1860) (IN) 2023-04-27 WO disclosed
WO-2023067628-A1 A METHOD FOR THE PREPARATION OF INDOLE-3-CARBOXYLIC ACID DERIVATIVES COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH AN INDIAN REGISTERED BODY INCORPORATED UNDER THE REGN. OF SOC. ACT (ACT XXI OF 1860) (IN) 2023-04-27 WO disclosed
EP-3288933-B1 OXINDOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF MUSC FOUND FOR RES DEV (US) 2021-10-06 EP disclosed
US-10370328-B2 Oxindole compounds and pharmaceutical compositions thereof MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2019-08-06 US disclosed
US-10253035-B2 Eis inhibitors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2019-04-09 US disclosed
US-20180162867-A1 EIS INHIBITORS UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION 2018-06-14 US disclosed
US-20180134659-A1 OXINDOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF MUSC FOUNDATION FOR RESEARCH DEVELOPMENT 2018-05-17 US disclosed
US-9920029-B2 Isatin compounds, compositions and methods for treatment of degenerative diseases and disorders MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2018-03-20 US disclosed
US-20100311715-A1 ALPHA CARBOLINES AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-12-09 US disclosed
US-7812018-B2 inhibitors of I kappa B kinase ( IKK-2) 2-amino-9-methyl-9H-pyrido[2,3-b]indole-3-carboxamide, useful for treating inflammatory diseases and cancer MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed
US-7812018-B2 inhibitors of I kappa B kinase ( IKK-2) 2-amino-9-methyl-9H-pyrido[2,3-b]indole-3-carboxamide, useful for treating inflammatory diseases and cancer MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed
US-7812018-B2 inhibitors of I kappa B kinase ( IKK-2) 2-amino-9-methyl-9H-pyrido[2,3-b]indole-3-carboxamide, useful for treating inflammatory diseases and cancer MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed
EP-1989203-A2 ALPHA CARBOLINES AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-11-12 EP disclosed
US-20070207997-A1 Alpha carbolines and uses thereof MILLENNIUM PHARMACEUTICALS, INC. 2007-09-06 US disclosed
US-20070207997-A1 Alpha carbolines and uses thereof MILLENNIUM PHARMACEUTICALS, INC. 2007-09-06 US disclosed
US-20070207997-A1 Alpha carbolines and uses thereof MILLENNIUM PHARMACEUTICALS, INC. 2007-09-06 US disclosed
WO-2007097981-A2 ALPHA CARBOLINES AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-08-30 WO disclosed
WO-2007097981-A2 ALPHA CARBOLINES AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-08-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11858915-B2 Polo like kinase 4 inhibitors PLK4, PLK2, PLK3 PARK7 1996/4885ALDH1A1 2211/4885ACHE 4244/4885
US-20250236590-A1 A METHOD FOR THE PREPARATION OF INDOLE-3-CARBOXYLIC ACID DERIVATIVES IDO1, INMT, IDO2 PARK7 1380/4885ALDH1A1 608/4885ACHE 101/4885
US-20180162867-A1 EIS INHIBITORS EP300, ACAT1, ACAT2 PARK7 4093/4885ALDH1A1 1232/4885ACHE 892/4885
US-10253035-B2 Eis inhibitors EP300, ACAT1, ACAT2 PARK7 4093/4885ALDH1A1 1232/4885ACHE 892/4885
US-20070207997-A1 Alpha carbolines and uses thereof CHRM1, CNR1, CXCR1 PARK7 58/4885ALDH1A1 416/4885ACHE 457/4885
US-10370328-B2 Oxindole compounds and pharmaceutical compositions thereof PARK7, OPRK1, COMT PARK7 1/4885ALDH1A1 212/4885ACHE 78/4885
US-20100311715-A1 ALPHA CARBOLINES AND USES THEREOF CHRM1, CNR1, CXCR1 PARK7 58/4885ALDH1A1 416/4885ACHE 457/4885
US-20180134659-A1 OXINDOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF PARK7, OPRK1, COMT PARK7 1/4885ALDH1A1 212/4885ACHE 78/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.