SCHEMBL3971374

SCHEMBL3971374

NC(=S)S.NCCCCCCNCCCCCCN.[NH2-].[Na+]

nearest known ligand 0.61

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 known ✓ O43570 2/20 0.54
CA2 known ✓ P00918 2/20 0.54
CA4 known ✓ P22748 2/20 0.54
CA1 known ✓ P00915 1/20 0.54
F13A1 P00488 2/20 0.54
CYP1A2 P05177 2/20 0.54
ALOX15 P16050 2/20 0.54
CA6 P23280 2/20 0.54
CA5A P35218 2/20 0.54
THPO P40225 2/20 0.54
CA7 P43166 2/20 0.54
CA9 Q16790 2/20 0.54
CA14 Q9ULX7 2/20 0.54
CA5B Q9Y2D0 2/20 0.54
CA3 P07451 1/20 0.54
CYP2C9 P11712 1/20 0.54
PKM P14618 1/20 0.54
TSHR P16473 1/20 0.54
MTOR P42345 1/20 0.54
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3967669 0.84 CA12 (0.55) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL11171595 0.81 CA12 (0.59) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL10336116 0.81 CA12 (0.59) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL31426982 0.81 DNM1 (0.53) CA12CA2CYP1A2ALOX15CA4
SCHEMBL28920597 0.79 CA12 (0.61) CA12F13A1CA2CYP1A2ALOX15
Trientine SCHEMBL29003404 0.79 CA12 (0.61) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL12983201 0.78 CA12 (0.87) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL5078139 0.78 CA12 (0.87) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL9182483 0.78 CA12 (0.87) CA12F13A1CA2CYP1A2ALOX15
SCHEMBL16295924 0.78 CA12 (0.87) CA12F13A1CA2CYP1A2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1302493-B1 Polydithiocarbamate resin AKZO NOBEL NV (NL) 2009-07-29 EP disclosed
US-7030205-B2 Polydithiocarbamate resin NATIONAL STARCH AND CHEMICAL INVESTMENT HOLDING CORPORATION (US) 2006-04-18 US disclosed
US-20030083456-A1 Polydithiocarbamate resin AKZO NOBEL N.V. (NL) 2003-05-01 US disclosed
EP-1302493-A2 Polydithiocarbamate resin National Starch and Chemical Investment Holding Corporation (US) 2003-04-16 EP disclosed