SCHEMBL3986249

SCHEMBL3986249

CCOC(=O)COc1ncc(Cl)c2cc(C)c(Cc3ccc(Cl)cc3)c(C)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.40
P2RX3 P56373 3/20 0.39
KDM4E B2RXH2 4/20 0.37
MAPT P10636 4/20 0.37
KMT2A Q03164 4/20 0.37
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
LMNA P02545 2/20 0.35
KCNH2 Q12809 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX5 P09917 1/20 0.35
OPRK1 P41145 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
RAB9A P51151 1/20 0.34
PPARG P37231 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3983780 0.89 THRB (0.46) HTTKDM4ETDP1ALOX5PPARG
SCHEMBL3984196 0.81 MAPT (0.41) HTTP2RX3KDM4EMAPTKMT2A
SCHEMBL11460802 0.70 NPSR1 (0.57) HTTP2RX3MAPTPOLBTDP1
SCHEMBL3985274 0.69 PTGDR2 (0.43) KDM4EMAPTKMT2AALDH1A1MEN1
SCHEMBL3345503 0.69 P2RX3 (0.42) P2RX3KDM4EMAPTKMT2AALDH1A1
SCHEMBL5494773 0.68 KDM4E (0.45) HTTKDM4EMAPTKMT2AALDH1A1
SCHEMBL3989733 0.68 LMNA (0.39) KDM4EKMT2AALDH1A1POLBTDP1
SCHEMBL3345008 0.68 P2RX3 (0.43) P2RX3KDM4EMAPTKMT2AALDH1A1
SCHEMBL3980177 0.66 DAO (0.43) KDM4EMAPTKMT2AALDH1A1MEN1
SCHEMBL3986256 0.66 TDP1 (0.43) HTTKDM4EMAPTTDP1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009060209-A1 6,6-FUSED BICYCLIC AROMATIC COMPOUNDS AND THEIR THERAPEUTI USE ARGENTA DISCOVERY LIMITED (GB) 2009-05-14 WO disclosed