SCHEMBL4023960

SCHEMBL4023960

CC(=O)Cc1ccc(O)c(C)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.61
ESR2 Q92731 4/20 0.61
GAA P10253 4/20 0.47
TDP1 Q9NUW8 3/20 0.47
TSHR P16473 2/20 0.47
NFKB1 P19838 2/20 0.47
POLB P06746 2/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
HPGD P15428 2/20 0.47
BLM P54132 2/20 0.47
HIF1A Q16665 2/20 0.47
HSD17B10 Q99714 2/20 0.47
RGS12 O14924 1/20 0.47
APEX1 P27695 1/20 0.47
THPO P40225 1/20 0.47
GNAI1 P63096 1/20 0.47
PMP22 Q01453 1/20 0.47
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28492275 0.86 ESR1 (0.63) ESR1ESR2GAATDP1TSHR
SCHEMBL30523685 0.84 HPGD (0.68) ESR1ESR2GAATDP1TSHR
SCHEMBL1362192 0.84 HPGD (0.68) ESR1ESR2GAATDP1TSHR
SCHEMBL12900623 0.83 LMNA (0.46) GAAPOLBLMNAALDH1A1
SCHEMBL1070431 0.83 KDM4E (0.67) ESR1GAATDP1TSHRNFKB1
SCHEMBL27907765 0.83 KDM4E (0.67) ESR1GAATDP1TSHRNFKB1
SCHEMBL23276708 0.82 ESR1 (0.59) ESR1ESR2GAATDP1TSHR
SCHEMBL2796509 0.82 ESR1 (0.59) ESR1ESR2GAATDP1TSHR
SCHEMBL1696094 0.81 ESR1 (0.57) ESR1ESR2TDP1KDM4ELMNA
SCHEMBL8733751 0.81 ESR1 (0.57) ESR1ESR2GAATDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701949-B1 ASSAY FOR ENTACTOGENS SIEMENS HEALTHCARE DIAGNOSTICS INC (US) 2018-04-18 EP disclosed
EP-2900654-A1 TETRAZOLINONE COMPOUNDS AND THEIR USE AS PESTICIDES Sumitomo Chemical Company Limited (JP) 2015-08-05 EP disclosed
US-8765809-B2 Ester derivative and use thereof AJINOMOTO CO., INC. (JP) 2014-07-01 US disclosed
EP-1701948-B1 ASSAY FOR ENTACTOGENS SIEMENS HEALTHCARE DIAGNOSTICS (US) 2014-03-26 EP disclosed
US-20130053441-A1 NOVEL ESTER DERIVATIVE AND USE THEREOF AJINOMOTO CO., INC. (JP) 2013-02-28 US disclosed
EP-1701948-A4 ASSAY FOR ENTACTOGENS SIEMENS HEALTHCARE DIAGNOSTICS (US) 2009-03-04 EP disclosed
WO-2008154023-A1 NOVEL USES OF PPAR DELTA AGONISTS CERENIS THERAPEUTICS S.A. (FR) 2008-12-18 WO disclosed
EP-1701949-A4 ASSAY FOR ENTACTOGENS DADE BEHRING INC (US) 2008-02-20 EP disclosed
EP-1863772-A1 AMIDE DERIVATIVES AS PPAR ACTIVATORS F.HOFFMANN-LA ROCHE AG (CH) 2007-12-12 EP disclosed
WO-2007028424-A1 AMIDE DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2007-03-15 WO disclosed
EP-1701948-A1 ASSAY FOR ENTACTOGENS DADE BEHRING INC. (US) 2006-09-20 EP disclosed
EP-1701949-A2 ASSAY FOR ENTACTOGENS DADE BEHRING INC. (US) 2006-09-20 EP disclosed
US-6991911-B2 Assay for entactogens DADE BEHRING INC. (US) 2006-01-31 US disclosed
WO-2005058864-A1 ASSAY FOR ENTACTOGENS DADE BEHRING INC. (US) 2005-06-30 WO disclosed
WO-2005058865-A2 ASSAY FOR ENTACTOGENS DADE BEHRING INC. (US) 2005-06-30 WO disclosed
US-20050130243-A1 Assay for entactogens SIEMENS HEALTHCARE DIAGNOSTICS INC. 2005-06-16 US disclosed
US-20050130244-A1 for detection of 3,4-methylenedioxyamphetamine (MDA), 3,4-methylenedioxy-methamphetamine (MDMA) anibody production; drug screening; haptens; immunogens SIEMENS HEALTHCARE DIAGNOSTICS INC. 2005-06-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130053441-A1 NOVEL ESTER DERIVATIVE AND USE THEREOF MEP1A, CES2, MEP1B ESR1 14/4885ESR2 122/4885GAA 3440/4885
US-20050130243-A1 Assay for entactogens HTR3C, COMT, PNMT ESR1 1577/4885ESR2 1926/4885GAA 898/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.