Puromycin

Puromycin

SCHEMBL4030642

COc1ccc(C[C@H](N)C(=O)NC2[C@@H](O)[C@H](n3cnc4c(N(C)C)ncnc43)O[C@@H]2CO)cc1.[Cl-].[Cl-].[H+].[H+]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Puromycin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPEPPS P55786 12/20 0.97
ANPEP P15144 10/20 0.97
SMN1; SMN2 Q16637 3/20 0.97
TP53 P04637 2/20 0.97
CYP3A4 P08684 2/20 0.97
LMNA P02545 1/20 0.97
HIF1A Q16665 1/20 0.97
HTT P42858 1/20 0.96
NPC1 O15118 1/20 0.96
RAB9A P51151 1/20 0.96
PAX8 Q06710 1/20 0.96
SLC29A1 Q99808 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Puromycin SCHEMBL14583797 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL3042415 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL21481061 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL14583945 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL22409382 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL24206459 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL22348910 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL20815730 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL21306559 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4
Puromycin SCHEMBL20393806 0.99 NPEPPS (1.00) NPEPPSANPEPSMN1; SMN2TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 76 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260102359-A1 COMBINATION TREATMENT OF DERMAL AND TRANSDERMAL FIBROTIC DISEASES, DISORDERS AND ASSOCIATED PAIN AND INFLAMMATION ERESINA LLC (US) 2026-04-16 US disclosed
EP-3259597-B2 PVRIG POLYPEPTIDES AND METHODS OF TREATMENT COMPUGEN LTD (IL) 2026-04-15 EP disclosed
US-20260069693-A1 UROLITHINS AND T-CELL MEDIATED IMMUNE RESPONSE CHEMOTHERAPEUTISCHES FORSCHUNGSINSTITUT GEORG SPEYER HAUS (DE) 2026-03-12 US disclosed
US-20250333503-A1 ANTI-PVRIG ANTIBODIES AND METHODS OF USE COMPUGEN LTD (IL) 2025-10-30 US disclosed
EP-4583863-A1 UROLITHINS AND T-CELL MEDIATED IMMUNE RESPONSE Chemotherapeutisches Forschungsinstitut Georg-Speyer-Haus (DE) 2025-07-16 EP disclosed
EP-4561556-A2 THERAPEUTIC USES OF UROLITHIN DERIVATIVES Vandria SA (CH) 2025-06-04 EP disclosed
US-12312404-B2 Anti-PVRIG antibodies and methods of use COMPUGEN LTD. (IL) 2025-05-27 US disclosed
CN-119947717-A Therapeutic use of urolithin derivatives 范徳利亚股份公司 2025-05-06 CN disclosed
CN-119120588-B Construction method of KCNB1 ion channel stable transgenic cell strain and application of KCNB1 ion channel stable transgenic cell strain in toxicity screening of plastic movable substances and degradation products 广州市华代生物科技有限公司 2025-02-28 CN disclosed
CN-119120384-B Cell strain stably transferring TRPA1 ion channel, construction method thereof and application thereof in screening of pain caused by immigrants of degradable material 广州市华代生物科技有限公司 2025-02-28 CN disclosed
US-20170029504-A1 ANTI-PVRIG ANTIBODIES AND METHODS OF USE COMPUGEN LTD. (IL) 2017-02-02 US disclosed
WO-2016134333-A9 ANTI-PVRIG ANTIBODIES AND METHODS OF USE COMPUGEN LTD. (IL) 2017-02-02 WO disclosed
WO-2016134335-A9 PVRIG POLYPEPTIDES AND METHODS OF TREATMENT COMPUGEN LTD. (IL) 2016-10-13 WO disclosed
WO-2016134333-A1 ANTI-PVRIG ANTIBODIES AND METHODS OF USE COMPUGEN LTD. (IL) 2016-08-25 WO disclosed
WO-2016134335-A2 PVRIG POLYPEPTIDES AND METHODS OF TREATMENT COMPUGEN LTD. (IL) 2016-08-25 WO disclosed
US-20160244521-A1 ANTI-PVRIG ANTIBODIES AND METHODS OF USE COMPUGEN LTD. (IL) 2016-08-25 US disclosed
US-9273364-B2 Transgenic reporter system that reveals expression profiles and regulation mechanisms of alternative splicing in mammalian organisms KYOTO UNIVERSITY (JP) 2016-03-01 US disclosed
US-20130137099-A1 TRANSGENIC REPORTER SYSTEM THAT REVEALS EXPRESSION PROFILES AND REGULATION MECHANISMS OF ALTERNATIVE SPLICING IN MAMMALIAN ORGANISMS KYOTO UNIVERSITY (JP) 2013-05-30 US disclosed
WO-2012113965-A1 METHOD FOR OBTAINING DATA THAT CAN BE USED TO EVALUATE, PREDICT AND/OR PROGNOSTICATE RESPONSE TO TREATMENT WITH PYRIMIDINE ANALOGUES SERVICIO ANDALUZ DE SALUD (ES) 2012-08-30 WO disclosed
WO-2009098451-A2 BIOMARKERS OF AMINOPEPTIDASE INHIBITION CHROMA THERAPEUTICS LIMITED (GB) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260069693-A1 UROLITHINS AND T-CELL MEDIATED IMMUNE RESPONSE MAVS, TFAM, MCU NPEPPS 4818/4885ANPEP 4531/4885SMN1; SMN2 1243/4885
US-20260102359-A1 COMBINATION TREATMENT OF DERMAL AND TRANSDERMAL FIBROTIC DISEASES, DISORDERS AND ASSOCIATED PAIN AND INFLAMMATION COL2A1, COLGALT1, PLOD3 NPEPPS 3071/4885ANPEP 3374/4885SMN1; SMN2 987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.