SCHEMBL4035489

SCHEMBL4035489

NC(=O)Oc1[nH]c2cccnc2c1Sc1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
TGFBR1 P36897 1/20 0.36
TGFBR2 P37173 1/20 0.36
PARP1 P09874 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHEK2 O96017 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035502 0.89 TUBB4A (0.39) SLC6A4PTGDR2ALDH1A1PARP1MEN1
SCHEMBL4032967 0.88 SMN1; SMN2 (0.41) SLC6A4PTGDR2ALDH1A1CYP1A2CYP3A4
SCHEMBL4033192 0.88 PKN1 (0.38) PARP1MEN1KMT2ACHEK2
SCHEMBL4036827 0.88 KDM4E (0.43) KDM4EALDH1A1HPGDTGFBR1TGFBR2
SCHEMBL4042064 0.84 TGFBR1 (0.38) KDM4EALDH1A1CYP3A4HPGDTGFBR1
SCHEMBL4033692 0.84 RHEB (0.42) ALDH1A1TGFBR1TGFBR2L3MBTL1RAB9A
SCHEMBL4039619 0.84 MAPT (0.46) KDM4EALDH1A1HPGDPARP1L3MBTL1
SCHEMBL4034008 0.83 LMNA (0.37) TGFBR1TGFBR2PARP1KMT2ALMNA
SCHEMBL4034813 0.83 PKM (0.43) KDM4EALDH1A1CYP3A4HPGDTGFBR1
SCHEMBL2053450 0.82 SLC6A4 (0.45) SLC6A4PTGDR2KDM4EALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed