SCHEMBL4033157

SCHEMBL4033157

NC(=O)NC=O.O=S(=O)(c1ccccc1)N1CCN(c2ccccc2-c2ccccc2)CC1C1CCc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.37
RAB9A P51151 3/20 0.37
HTR1A P08908 3/20 0.37
NPC1 O15118 1/20 0.37
MTOR P42345 1/20 0.37
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALDH1A1 P00352 3/20 0.34
TSHR P16473 2/20 0.33
HSD11B1 P28845 1/20 0.33
DRD3 P35462 4/20 0.33
AKR1C3 P42330 1/20 0.33
HTR7 P34969 2/20 0.33
USP2 O75604 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4220008 0.86 ALDH1A1 (0.40) KMT2ANPSR1MAPTALDH1A1TSHR
SCHEMBL4037792 0.75 ALDH1A1 (0.37) DRD2HTR1ACYP2C19KMT2AMEN1
SCHEMBL4038524 0.71 MMP2 (0.34)
SCHEMBL6190430 0.66 MEN1 (0.42) CYP3A4CYP2C19KMT2ANPSR1MEN1
SCHEMBL4217064 0.65 FABP1 (0.42) NPSR1MAPTALDH1A1TSHRUSP2
SCHEMBL4223317 0.62 DRD2 (0.36) DRD2HTR1ACYP3A4ALDH1A1DRD3
SCHEMBL4036984 0.61 ALDH1A1 (0.47) KMT2AALDH1A1USP2
SCHEMBL6190434 0.61 GAA (0.48) KMT2ANPSR1MEN1ALDH1A1TSHR
SCHEMBL8163062 0.60 ALDH1A1 (0.52) HTR1ANPSR1MAPTALDH1A1TSHR
SCHEMBL4035867 0.60 CA1 (0.46) CYP3A4CYP2C19CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed