SCHEMBL4033612

SCHEMBL4033612

CCCCCc1ccc(C(=O)N2CCN(S(=O)(=O)c3ccc4ncccc4c3)C(C(=O)N3CCCCC3CO)C2)c(=O)o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.38
ALDH1A1 P00352 2/20 0.38
NR2F2 P24468 1/20 0.38
CHRM1 P11229 1/20 0.36
HTR7 P34969 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.33
NPC1 O15118 2/20 0.33
GALR3 O60755 1/20 0.32
ATM Q13315 1/20 0.32
LMNA P02545 1/20 0.32
ABL1 P00519 1/20 0.32
RIN1 Q13671 1/20 0.32
KDM2B Q8NHM5 1/20 0.32
HPGD P15428 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
ADRB2 P07550 1/20 0.32
KMT2A Q03164 1/20 0.32
SMO Q99835 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033608 0.87 ALOX15 (0.41) ALDH1A1HPGDMAPTHTTKMT2A
SCHEMBL4035745 0.81 MMP1 (0.40) ALDH1A1CHRM1
SCHEMBL4037876 0.81 ALDH1A1 (0.46) ALDH1A1CHRM1HPGDHTTKMT2A
SCHEMBL6209492 0.79 ALOX15 (0.41) ALDH1A1HPGDMAPTHTTKMT2A
SCHEMBL4034716 0.79 P2RX7 (0.42)
SCHEMBL4033601 0.76 TP53 (0.40) ALDH1A1LMNAMAPTHTTKMT2A
SCHEMBL7090151 0.74 EPHX2 (0.41) RAB9AALDH1A1NR2F2NPC1MAPT
SCHEMBL1386085 0.68 MAPK1 (0.51) ALDH1A1ATMLMNAHPGDMAPT
SCHEMBL1381941 0.68 PKM (0.54) ALDH1A1ATMHPGDMAPTKMT2A
SCHEMBL4034713 0.67 ALDH1A1 (0.44) ALDH1A1ATMLMNAHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed