SCHEMBL4037876

SCHEMBL4037876

CCCCCc1ccc(C(=O)N2CCN(S(=O)(=O)c3ccc4ncccc4c3)C(C(=O)NCc3ccco3)C2)c(=O)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.46
USP2 O75604 1/20 0.46
KDM4E B2RXH2 1/20 0.44
PKM P14618 3/20 0.40
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP9 P14780 1/20 0.36
MMP13 P45452 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
CHRM1 P11229 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035745 0.91 MMP1 (0.40) ALDH1A1USP2KDM4EMMP1MMP3
SCHEMBL4034716 0.88 P2RX7 (0.42)
SCHEMBL1381941 0.87 PKM (0.54) ALDH1A1USP2PKMSMN1; SMN2KMT2A
SCHEMBL4033612 0.81 RAB9A (0.38) ALDH1A1KMT2AHTTCHRM1HPGD
SCHEMBL6209732 0.79 ALDH1A1 (0.45) ALDH1A1PKMKMT2AGAAHPGD
SCHEMBL1386085 0.78 MAPK1 (0.51) ALDH1A1PKMSMN1; SMN2KMT2AGAA
SCHEMBL4038385 0.78 ALDH1A1 (0.57) ALDH1A1USP2KDM4EPKMSMN1; SMN2
SCHEMBL4036566 0.77 ALDH1A1 (0.62) ALDH1A1USP2KDM4EPKMSMN1; SMN2
SCHEMBL4034713 0.76 ALDH1A1 (0.44) ALDH1A1PKMSMN1; SMN2HPGDMAPK1
SCHEMBL7090151 0.72 EPHX2 (0.41) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed