SCHEMBL4040800

SCHEMBL4040800

CCCC(NC(=O)Oc1oc2ccccc2c1C)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.36
FAP Q12884 2/20 0.36
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.32
CTSK P43235 14/20 0.31
CTSL P07711 12/20 0.31
CTSS P25774 8/20 0.31
CTSB P07858 3/20 0.31
CTSV O60911 2/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042095 0.93 CTSK (0.39) NPC1RAB9ASMN1; SMN2CTSKCTSL
SCHEMBL4047097 0.92 CTSL (0.33) NPC1RAB9ASMN1; SMN2TSHRCTSK
SCHEMBL4043247 0.90 CTSK (0.39) PREPFAPCTSKCTSLCTSS
SCHEMBL4045248 0.89 NPC1 (0.33) NPC1RAB9ASMN1; SMN2TSHRCTSK
SCHEMBL4048128 0.89 CHRNB2 (0.36) PREPFAPSMN1; SMN2TSHRGAA
SCHEMBL4040090 0.88 PREP (0.36) PREPFAPCTSKCTSLCTSS
SCHEMBL4048824 0.86 CTSK (0.37) PREPFAPNPC1RAB9ACTSK
SCHEMBL4042714 0.85 SMN1; SMN2 (0.36) PREPFAPSMN1; SMN2TSHRCTSK
SCHEMBL4044689 0.85 PREP (0.35) PREPFAPCTSKCTSLCTSS
SCHEMBL4050441 0.85 CTSK (0.39) PREPFAPNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed