SCHEMBL4041586

SCHEMBL4041586

NC(=O)C1C[N+](Cc2ccccc2)(C(=O)c2ccccc2)CCN1S(=O)(=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 4/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA9 Q16790 2/20 0.40
ALDH1A1 P00352 3/20 0.40
MMP1 P03956 4/20 0.38
MMP9 P14780 4/20 0.38
MMP13 P45452 4/20 0.38
MMP3 P08254 2/20 0.38
MMP7 P09237 2/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032958 0.88 ALDH1A1 (0.43) FKBP1AALDH1A1MMP1MMP9MMP13
SCHEMBL4038466 0.76 ALDH1A1 (0.43) FKBP1AALDH1A1MMP1MMP9MMP13
SCHEMBL4033188 0.75 ALDH1A1 (0.46) ALDH1A1
SCHEMBL4038075 0.72 ALDH1A1 (0.47) ALDH1A1NPSR1
SCHEMBL4036533 0.70 MMP3 (0.43) ALDH1A1MMP1MMP9MMP13MMP3
SCHEMBL695071 0.70 MMP2 (0.59) FKBP1AALDH1A1MMP9NPSR1
SCHEMBL17833176 0.70 MMP2 (0.59) FKBP1AALDH1A1MMP9NPSR1
SCHEMBL8718942 0.69 LMNA (0.58) FKBP1AALDH1A1MMP9MAPK1NPSR1
SCHEMBL4704780 0.67 ALDH1A1 (0.46) FKBP1AALDH1A1MMP9NPSR1
SCHEMBL14843813 0.66 MMP1 (0.52) ALDH1A1MMP1MMP9MMP13MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed