SCHEMBL4046868

SCHEMBL4046868

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.37
ITGAV P06756 1/20 0.37
KCNQ1 P51787 1/20 0.37
BCL2 P10415 2/20 0.36
ELOVL6 Q9H5J4 1/20 0.35
F2 P00734 1/20 0.35
ALDH1A1 P00352 2/20 0.35
NAMPT P43490 1/20 0.35
GPR132 Q9UNW8 1/20 0.34
CTSK P43235 3/20 0.34
ACE2 Q9BYF1 1/20 0.34
ITGA4 P13612 3/20 0.34
ITGB7 P26010 3/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CASP3 P42574 1/20 0.34
CASP7 P55210 1/20 0.34
CASP6 P55212 1/20 0.34
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041436 0.94 ALDH1A1 (0.39) ITGB1ITGAVKCNQ1BCL2F2
SCHEMBL4047882 0.93 F2 (0.36) ITGB1ITGAVKCNQ1BCL2ELOVL6
SCHEMBL4047615 0.90 CTSB (0.38) BCL2F2NAMPTGPR132CTSK
SCHEMBL4042529 0.90 BCL2 (0.38) BCL2GPR132CTSKITGA4ITGB7
SCHEMBL4046036 0.89 P2RX7 (0.36) ITGB1BCL2CTSKITGA4ITGB7
SCHEMBL4051777 0.89 CTSK (0.44) KCNQ1ELOVL6ALDH1A1NAMPTCTSK
SCHEMBL4048312 0.88 KCNQ1 (0.40) KCNQ1ELOVL6ALDH1A1NAMPTCTSK
SCHEMBL4041433 0.88 ALDH1A1 (0.35) ITGB1ITGAVF2ALDH1A1ITGA4
SCHEMBL4041003 0.87 CTSL (0.39) CTSKCTSBCTSS
SCHEMBL4049549 0.85 GPR132 (0.38) GPR132CTSKACE2ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed