SCHEMBL4043031

SCHEMBL4043031

CCCC(NC(=O)Oc1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 1/20 0.37
CTSK P43235 4/20 0.36
C3AR1 Q16581 1/20 0.36
DRD4 P21917 1/20 0.35
MC4R P32245 1/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35
ACACB O00763 1/20 0.35
PAX8 Q06710 1/20 0.35
TACR1 P25103 1/20 0.35
GPR132 Q9UNW8 3/20 0.34
CCR1 P32246 1/20 0.34
ROCK2 O75116 1/20 0.34
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34
NAMPT P43490 1/20 0.34
CHRNA7 P36544 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044443 0.93 ALDH1A1 (0.38) HTRA1CTSKACACBPAX8GPR132
SCHEMBL4045179 0.92 CTSK (0.44) HTRA1CTSKC3AR1DRD4PAX8
SCHEMBL4047771 0.91 CTSK (0.39) CTSKACACBGPR132CHRNA7
SCHEMBL4046542 0.89 POLB (0.36) CTSKACACBPAX8GPR132
SCHEMBL4041238 0.89 CHRNB2 (0.36) HTRA1CTSKMC4RMC3RMC1R
SCHEMBL4043616 0.89 CTSK (0.35) HTRA1CTSKPAX8TACR1GPR132
SCHEMBL4046786 0.88 CHRNB2 (0.36) HTRA1CTSKPAX8GPR132NAMPT
SCHEMBL4040981 0.87 CTSK (0.35) CTSKACACBPAX8GPR132CHRNA7
SCHEMBL4045728 0.87 CTSK (0.35) CTSKC3AR1ACACBPAX8GPR132
SCHEMBL4047844 0.87 SMYD3 (0.35) HTRA1CTSKC3AR1DRD4MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed