SCHEMBL4043383

SCHEMBL4043383

CCCC(NC(=O)Oc1cc2cc(OC)ccc2o1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 7/20 0.35
TAS1R1 Q7RTX1 7/20 0.35
BCAT1 P54687 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
F2 P00734 1/20 0.30
PRSS1 P07477 1/20 0.30
TP53 P04637 1/20 0.30
KCNQ1 P51787 1/20 0.30
ELOVL6 Q9H5J4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049248 0.93 CTSV (0.31) TAS1R3TAS1R1BCAT1ALDH1A1GAA
SCHEMBL4042354 0.93 TAS1R3 (0.37) TAS1R3TAS1R1BCAT1ALDH1A1GAA
SCHEMBL4051242 0.92 CTSK (0.33)
SCHEMBL4045162 0.90 TAS1R3 (0.34) TAS1R3TAS1R1F2
SCHEMBL6242334 0.90 TAS1R3 (0.46) TAS1R3TAS1R1BCAT1
SCHEMBL4044402 0.90 GAA (0.36) TAS1R3TAS1R1ALDH1A1GAAF2
SCHEMBL4043869 0.89 KCNQ1 (0.37) TAS1R3TAS1R1ALDH1A1KCNQ1ELOVL6
SCHEMBL4045579 0.87 HPGD (0.32) ALDH1A1
SCHEMBL4042533 0.86 CTSK (0.40)
SCHEMBL4045249 0.86 CTSK (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed