SCHEMBL4049248

SCHEMBL4049248

COc1ccc2oc(OC(=O)NC(CC3CC3)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)c3ccc[n+]([O-])c3)cc2c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.31
CTSL P07711 2/20 0.31
CTSS P25774 2/20 0.31
TAS1R3 Q7RTX0 2/20 0.31
TAS1R1 Q7RTX1 2/20 0.31
BCAT1 P54687 1/20 0.31
POLB P06746 2/20 0.31
L3MBTL1 Q9Y468 3/20 0.31
GAA P10253 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
F2 P00734 1/20 0.31
PRSS1 P07477 1/20 0.31
PTPN22 Q9Y2R2 1/20 0.31
TP53 P04637 1/20 0.31
KCNQ1 P51787 1/20 0.30
ATM Q13315 1/20 0.30
KDM4E B2RXH2 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042354 0.94 TAS1R3 (0.37) CTSVCTSLCTSSTAS1R3TAS1R1
SCHEMBL4043383 0.93 TAS1R3 (0.35) TAS1R3TAS1R1BCAT1L3MBTL1GAA
SCHEMBL4043929 0.91 CTSV (0.32) CTSVCTSLCTSSTAS1R3TAS1R1
SCHEMBL4044402 0.90 GAA (0.36) TAS1R3TAS1R1GAAALDH1A1F2
SCHEMBL4043537 0.90 PIK3CG (0.37) POLBALDH1A1LMNASMN1; SMN2KCNQ1
SCHEMBL4048699 0.87 CTSK (0.40) CTSVCTSLCTSS
SCHEMBL4042413 0.85 CTSK (0.40) CTSVCTSLCTSSTAS1R3TAS1R1
SCHEMBL4051242 0.84 CTSK (0.33) CTSVCTSLCTSS
SCHEMBL4050896 0.84 HPGD (0.34) CTSVCTSLCTSSGAAALDH1A1
SCHEMBL4045043 0.84 HPGD (0.38) CTSVCTSLCTSSPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed