SCHEMBL4044539

SCHEMBL4044539

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
ELANE P08246 1/20 0.34
CTSK P43235 3/20 0.34
ACE2 Q9BYF1 1/20 0.34
GPR132 Q9UNW8 1/20 0.33
ACE P12821 2/20 0.33
HDAC8 Q9BY41 1/20 0.33
P2RX7 Q99572 1/20 0.33
PRCP P42785 1/20 0.33
BCL2 P10415 1/20 0.33
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
XIAP P98170 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049324 0.94 MC4R (0.37) ITGA4ITGB7ELANECTSKP2RX7
SCHEMBL4051785 0.94 ITGA4 (0.39) ITGA4ITGB7ELANECTSKHDAC8
SCHEMBL4046932 0.93 GPR132 (0.35) ITGA4ITGB7FNTAFNTBELANE
SCHEMBL4041003 0.90 CTSL (0.39) CTSKCTSLCTSBCTSS
SCHEMBL4045311 0.89 CTSK (0.43) ELANECTSKCTSLCTSBCTSS
SCHEMBL4047615 0.88 CTSB (0.38) CTSKACE2GPR132ACEBCL2
SCHEMBL4043139 0.88 ELANE (0.37) ITGA4ITGB7ELANECTSK
SCHEMBL4045047 0.88 CTSL (0.37) ITGA4ITGB7FNTAFNTBCTSK
SCHEMBL4044814 0.88 FNTA (0.35) ITGA4ITGB7FNTAFNTBCTSK
SCHEMBL4048142 0.87 GAA (0.36) ITGA4ITGB7FNTAFNTBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed