SCHEMBL4044198

SCHEMBL4044198

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccccn1)Oc1cccc2cccnc12

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 13/20 0.42
CTSS P25774 13/20 0.42
CTSK P43235 13/20 0.42
CTSB P07858 6/20 0.39
CTSV O60911 2/20 0.38
CNR1 P21554 3/20 0.36
GAA P10253 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044768 0.93 CTSL (0.44) CTSLCTSSCTSKCTSBCTSV
SCHEMBL4048142 0.90 GAA (0.36) CTSLCTSSCTSKCTSBCNR1
SCHEMBL4040381 0.90 MC4R (0.36) CTSLCTSSCTSKCNR1GAA
SCHEMBL4041745 0.89 CNR1 (0.39) CTSLCTSSCTSKCNR1GAA
SCHEMBL4042222 0.88 CNR1 (0.34) CTSLCTSSCTSKCNR1GAA
SCHEMBL4044157 0.88 CNR1 (0.38) CTSLCTSSCTSKCNR1GAA
SCHEMBL4042762 0.87 GAA (0.34) CTSLCTSSCTSKCTSBCNR1
SCHEMBL4052351 0.86 CNR1 (0.36) CTSKCNR1GAAALDH1A1SMN1; SMN2
SCHEMBL4049994 0.86 CTSK (0.40) CTSLCTSSCTSKGAAALDH1A1
SCHEMBL4041003 0.86 CTSL (0.39) CTSLCTSSCTSKCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed