SCHEMBL4042762

SCHEMBL4042762

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)Oc1cccc2cccnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.34
CTSB P07858 1/20 0.34
CNR1 P21554 3/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
CTSL P07711 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
GPR132 Q9UNW8 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
ACE P12821 1/20 0.32
KDM4E B2RXH2 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPK1 P28482 1/20 0.32
F12 P00748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042676 0.92 CTSB (0.36) MAPTCTSSCTSKCTSBCTSL
SCHEMBL4041745 0.91 CNR1 (0.39) GAAMAPTNPSR1CTSSCTSK
SCHEMBL4048142 0.90 GAA (0.36) GAAMAPTNPSR1CTSSCTSK
SCHEMBL4052351 0.89 CNR1 (0.36) GAAMAPTNPSR1CTSKCNR1
SCHEMBL4044198 0.87 CTSL (0.42) GAAMAPTNPSR1CTSSCTSK
SCHEMBL4047615 0.86 CTSB (0.38) CTSSCTSKCTSBGPR132ACE
SCHEMBL4040381 0.85 MC4R (0.36) GAAMAPTNPSR1CTSSCTSK
SCHEMBL4044157 0.85 CNR1 (0.38) GAAMAPTNPSR1CTSSCTSK
SCHEMBL4045047 0.84 CTSL (0.37) GAAMAPTNPSR1CTSSCTSK
SCHEMBL4042222 0.84 CNR1 (0.34) GAAMAPTNPSR1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed