SCHEMBL4044157

SCHEMBL4044157

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1)Oc1cccc2cccnc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.38
L3MBTL1 Q9Y468 1/20 0.35
ITGA4 P13612 2/20 0.33
ITGB7 P26010 1/20 0.33
ALDH1A1 P00352 3/20 0.33
GAA P10253 2/20 0.33
MAPK1 P28482 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TSHR P16473 1/20 0.33
CNR2 P34972 1/20 0.33
ITGB1 P05556 1/20 0.33
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
MMP1 P03956 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041745 0.91 CNR1 (0.39) CNR1L3MBTL1ITGA4ITGB7ALDH1A1
SCHEMBL4045912 0.90 ITGA4 (0.34) ITGA4ITGB7ITGB1CTSLCTSS
SCHEMBL4042222 0.90 CNR1 (0.34) CNR1L3MBTL1ITGA4ALDH1A1GAA
SCHEMBL4044198 0.88 CTSL (0.42) CNR1ALDH1A1GAAMAPK1SMN1; SMN2
SCHEMBL4048142 0.85 GAA (0.36) CNR1L3MBTL1ITGA4ITGB7ALDH1A1
SCHEMBL4040381 0.85 MC4R (0.36) CNR1ITGA4ALDH1A1GAAMAPT
SCHEMBL4042762 0.85 GAA (0.34) CNR1L3MBTL1ALDH1A1GAAMAPK1
SCHEMBL4052351 0.84 CNR1 (0.36) CNR1L3MBTL1ITGA4ALDH1A1GAA
SCHEMBL4046036 0.84 P2RX7 (0.36) ITGA4ITGB7ITGB1CTSK
SCHEMBL4041433 0.83 ALDH1A1 (0.35) ITGA4ITGB7ALDH1A1TSHRITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed