SCHEMBL4041745

SCHEMBL4041745

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1)Oc1cccc2cccnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.39
L3MBTL1 Q9Y468 1/20 0.36
ITGB1 P05556 2/20 0.34
ITGAV P06756 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ITGA4 P13612 2/20 0.34
ITGB7 P26010 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 2/20 0.33
GAA P10253 2/20 0.33
TSHR P16473 2/20 0.33
CNR2 P34972 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALOX15 P16050 1/20 0.33
CTSL P07711 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
CASP3 P42574 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041433 0.92 ALDH1A1 (0.35) ITGB1ITGAVHSD17B10ITGA4ITGB7
SCHEMBL4044157 0.91 CNR1 (0.38) CNR1L3MBTL1ITGB1ITGA4ITGB7
SCHEMBL4042762 0.91 GAA (0.34) CNR1L3MBTL1ALDH1A1MAPK1GAA
SCHEMBL4052351 0.90 CNR1 (0.36) CNR1L3MBTL1ITGB1ITGA4ALDH1A1
SCHEMBL4044198 0.89 CTSL (0.42) CNR1ALDH1A1MAPK1GAATSHR
SCHEMBL4040381 0.86 MC4R (0.36) CNR1ITGB1ITGA4ALDH1A1GAA
SCHEMBL4048142 0.86 GAA (0.36) CNR1L3MBTL1HSD17B10ITGA4ITGB7
SCHEMBL4042222 0.86 CNR1 (0.34) CNR1L3MBTL1ITGB1ITGA4ALDH1A1
SCHEMBL4046868 0.85 ITGB1 (0.37) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL4042676 0.83 CTSB (0.36) L3MBTL1ALDH1A1MAPK1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed