SCHEMBL4042222

SCHEMBL4042222

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccc[n+]1[O-])Oc1cccc2cccnc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.34
GAA P10253 3/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TSHR P16473 1/20 0.33
CTSL P07711 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 2/20 0.33
HPGD P15428 1/20 0.33
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
FABP1 P07148 1/20 0.32
HSP90AA1 P07900 1/20 0.32
TP53 P04637 1/20 0.32
CNR2 P34972 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045610 0.91 POLB (0.33) CTSLCTSSCTSK
SCHEMBL4044157 0.90 CNR1 (0.38) CNR1GAAMAPTNPSR1TSHR
SCHEMBL4044198 0.88 CTSL (0.42) CNR1GAAMAPTNPSR1TSHR
SCHEMBL4041745 0.86 CNR1 (0.39) CNR1GAAMAPTNPSR1TSHR
SCHEMBL4040381 0.85 MC4R (0.36) CNR1GAAMAPTNPSR1TSHR
SCHEMBL4048142 0.85 GAA (0.36) CNR1GAAMAPTNPSR1TSHR
SCHEMBL4047239 0.84 CTSK (0.34) CTSK
SCHEMBL4042762 0.84 GAA (0.34) CNR1GAAMAPTNPSR1CTSL
SCHEMBL4052351 0.83 CNR1 (0.36) CNR1GAAMAPTNPSR1CTSK
SCHEMBL6211991 0.82 CTSL (0.40) CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed