SCHEMBL4042165

SCHEMBL4042165

O=C(NC(Cc1cccc(O)c1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
CTSK P43235 3/20 0.37
ACE P12821 2/20 0.36
GPR132 Q9UNW8 5/20 0.36
CHRNA7 P36544 1/20 0.36
CMKLR2 P46091 1/20 0.36
CMKLR1 Q99788 1/20 0.36
CTSB P07858 3/20 0.35
CTSS P25774 3/20 0.35
CTSL P07711 2/20 0.35
ECE1 P42892 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
CTSV O60911 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049549 0.93 GPR132 (0.38) EPHX1CTSKACEGPR132CHRNA7
SCHEMBL6209046 0.90 CTSK (0.47) CTSKACEGPR132CMKLR2CMKLR1
SCHEMBL4040214 0.90 GPR132 (0.39) CTSKACEGPR132CHRNA7ECE1
SCHEMBL4041149 0.90 ITGA4 (0.39) CTSKACECHRNA7ECE1
SCHEMBL4045083 0.88 CTSK (0.47) EPHX1CTSKCHRNA7CTSBCTSS
SCHEMBL4047771 0.87 CTSK (0.39) EPHX1CTSKGPR132CHRNA7ECE1
SCHEMBL4044160 0.87 CTSB (0.37) EPHX1CTSKACEGPR132CHRNA7
SCHEMBL4047882 0.86 F2 (0.36) EPHX1CTSKACEGPR132CHRNA7
SCHEMBL4045597 0.85 ACE (0.36) EPHX1CTSKACEGPR132CHRNA7
SCHEMBL4045030 0.85 CTSK (0.41) CTSKACEGPR132CTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed