SCHEMBL4045552

SCHEMBL4045552

COc1ccc(CC(NC(=O)Oc2ccc(-c3ccccc3)cc2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)c2cccc[n+]2[O-])cc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
HDAC8 Q9BY41 1/20 0.35
CTSK P43235 3/20 0.35
ITGA4 P13612 6/20 0.35
ITGB7 P26010 5/20 0.35
ITGB1 P05556 2/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 1/20 0.34
P2RX7 Q99572 1/20 0.34
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
ADAM17 P78536 1/20 0.34
BCL2 P10415 1/20 0.34
TSHR P16473 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047239 0.94 CTSK (0.34) CTSKP2RX7
SCHEMBL4047305 0.93 P2RX7 (0.37) CTSKITGA4ITGB7ITGB1P2RX7
SCHEMBL4041712 0.90 ITGA4 (0.40) ITGB3ITGAVHDAC8CTSKITGA4
SCHEMBL4047763 0.89 CTSK (0.44) CTSKKMT2A
SCHEMBL4047214 0.89 CTSK (0.33) ITGB3ITGAVCTSKITGA4ITGB1
SCHEMBL4041133 0.89 CTSK (0.36) CTSK
SCHEMBL4039714 0.86 CTSK (0.51) CTSKKMT2ACA2
SCHEMBL4046036 0.84 P2RX7 (0.36) CTSKITGA4ITGB7ITGB1P2RX7
SCHEMBL6234334 0.84 CTSK (0.44) ITGB3CTSKITGA4ITGB1KMT2A
SCHEMBL4041901 0.83 P2RX7 (0.39) CTSKITGA4ITGB7ITGB1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed