SCHEMBL4046036

SCHEMBL4046036

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.36
ITGA4 P13612 5/20 0.36
ITGB7 P26010 4/20 0.36
BCL2 P10415 1/20 0.35
CTSK P43235 3/20 0.35
ITGB1 P05556 2/20 0.35
ACE P12821 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041712 0.94 ITGA4 (0.40) ITGA4ITGB7BCL2CTSKITGB1
SCHEMBL4041901 0.94 P2RX7 (0.39) P2RX7ITGA4ITGB7CTSKITGB1
SCHEMBL4043833 0.92 F10 (0.36) P2RX7ITGA4ITGB7CTSKITGB1
SCHEMBL4047239 0.90 CTSK (0.34) P2RX7CTSKACE
SCHEMBL4046868 0.89 ITGB1 (0.37) P2RX7ITGA4ITGB7BCL2CTSK
SCHEMBL4045912 0.88 ITGA4 (0.34) P2RX7ITGA4ITGB7CTSKITGB1
SCHEMBL4044695 0.88 CTSK (0.36) CTSK
SCHEMBL4041003 0.86 CTSL (0.39) CTSK
SCHEMBL4045552 0.84 ITGB3 (0.37) P2RX7ITGA4ITGB7BCL2CTSK
SCHEMBL4047305 0.84 P2RX7 (0.37) P2RX7ITGA4ITGB7CTSKITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2016064-A2 METHODS FOR THE PREPARATION OF PYRAZOLE-CONTAINING COMPOUNDS Janssen Pharmaceutica, N.V. (BE) 2009-01-21 EP claimed
WO-2007131153-A2 METHODS FOR THE PREPARATION OF PYRAZOLE-CONTAINING COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2007-11-15 WO claimed