SCHEMBL4047214

SCHEMBL4047214

O=C(NC(Cc1cccc(O)c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccc[n+]1[O-])Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.33
P2RX7 Q99572 5/20 0.32
HPGDS O60760 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
F10 P00742 2/20 0.31
F2 P00734 1/20 0.31
PLG P00747 1/20 0.31
ST14 Q9Y5Y6 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGAV P06756 1/20 0.31
ADAMTS4 O75173 1/20 0.31
MMP13 P45452 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047239 0.93 CTSK (0.34) CTSKP2RX7OPRM1
SCHEMBL4043833 0.91 F10 (0.36) CTSKP2RX7ITGB1ITGA4F10
SCHEMBL4047305 0.89 P2RX7 (0.37) CTSKP2RX7ITGB1ITGA4
SCHEMBL4045552 0.89 ITGB3 (0.37) CTSKP2RX7ITGB1ITGA4ITGB3
SCHEMBL4047763 0.87 CTSK (0.44) CTSK
SCHEMBL4041133 0.86 CTSK (0.36) CTSKF10F2
SCHEMBL4051296 0.85 CTSL (0.39) CTSK
SCHEMBL4047882 0.84 F2 (0.36) CTSKITGB1F10F2PLG
SCHEMBL4047934 0.83 CTSK (0.51) CTSKHPGDSF10PLGITGB3
SCHEMBL4046036 0.83 P2RX7 (0.36) CTSKP2RX7ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed