SCHEMBL4041712

SCHEMBL4041712

COc1ccc(CC(NC(=O)Oc2ccc(-c3ccccc3)cc2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)c2ccc[n+]([O-])c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 8/20 0.40
ITGB7 P26010 8/20 0.40
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
PLG P00747 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38
BCL2 P10415 1/20 0.37
MMP1 P03956 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
KCNQ1 P51787 2/20 0.37
ITGB1 P05556 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046036 0.94 P2RX7 (0.36) ITGA4ITGB7BCL2ITGB1CTSK
SCHEMBL4041901 0.93 P2RX7 (0.39) ITGA4ITGB7ITGB1CTSK
SCHEMBL4045552 0.90 ITGB3 (0.37) ITGA4ITGB7ITGB3ITGAVBCL2
SCHEMBL4043833 0.89 F10 (0.36) ITGA4ITGB7F2F10PLG
SCHEMBL4044695 0.88 CTSK (0.36) MMP1MMP3MMP7MMP9MMP13
SCHEMBL4048167 0.85 CTSK (0.50) F2F10PLGST14KMT2A
SCHEMBL4047239 0.84 CTSK (0.34) CTSK
SCHEMBL4047305 0.83 P2RX7 (0.37) ITGA4ITGB7ITGB1CTSK
SCHEMBL4045924 0.83 USP30 (0.40) ITGA4ITGB7ITGB3ITGAVITGB1
SCHEMBL4051785 0.83 ITGA4 (0.39) ITGA4ITGB7ITGB3ITGAVMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed