SCHEMBL4056098

SCHEMBL4056098

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)CNS(=O)(=O)c1cnc(Cl)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.35
ALDH1A1 P00352 2/20 0.33
CYP51A1 Q16850 1/20 0.33
HTRA1 Q92743 1/20 0.33
STAT6 P42226 1/20 0.33
HTT P42858 1/20 0.32
BCAT1 P54687 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
PYGL P06737 1/20 0.32
HSPA5 P11021 1/20 0.32
HSPA8 P11142 1/20 0.32
HSPA9 P38646 1/20 0.32
HSPA2 P54652 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4057362 0.83 PYGL (0.39) DRD2CYP51A1BCAT1PYGL
SCHEMBL4057673 0.83 PYGL (0.39) DRD2CYP51A1STAT6BCAT1PYGL
SCHEMBL4049377 0.81 CYP51A1 (0.39) DRD2CYP51A1STAT6PYGL
SCHEMBL4050835 0.81 DRD2 (0.39) DRD2CYP51A1STAT6PYGL
SCHEMBL4052196 0.81 DRD4 (0.38) DRD2CYP51A1STAT6PYGL
SCHEMBL4050168 0.81 DRD2 (0.36) DRD2ALDH1A1CYP51A1STAT6PYGL
SCHEMBL19856906 0.79 DRD2 (0.45) DRD2ALDH1A1CYP51A1STAT6PYGL
SCHEMBL4051117 0.78 ALOX15 (0.42) CYP51A1BCAT1PYGL
SCHEMBL1550540 0.76 DRD2 (0.40) DRD2CYP51A1HTRA1STAT6HSPA5
SCHEMBL7983935 0.76 DRD2 (0.35) DRD2ALDH1A1CYP51A1BCAT1PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO claimed
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed