SCHEMBL4050322

SCHEMBL4050322

CCCC(NC(=O)Oc1cccs1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.34
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
PREP P48147 3/20 0.32
FAP Q12884 2/20 0.32
ALDH1A1 P00352 1/20 0.32
ELANE P08246 1/20 0.31
KMT2A Q03164 1/20 0.31
DHPS P49366 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049412 0.92 CTSK (0.42) CTSKMAPK1CYP2C19PREPFAP
SCHEMBL4042699 0.89 CTSK (0.32) CTSKPREPFAP
SCHEMBL4047006 0.89 HSD17B10 (0.38) CTSKALDH1A1
SCHEMBL4045553 0.89 CTSK (0.34) CTSKPREPFAPALDH1A1ELANE
SCHEMBL4044808 0.88 CTSK (0.36) CTSKPREPFAPELANE
SCHEMBL4042570 0.88 CTSK (0.34) CTSKPREPFAPALDH1A1ELANE
SCHEMBL4050153 0.88 SMYD3 (0.35) CYP2C19ALDH1A1
SCHEMBL4043596 0.88 ELANE (0.38) CTSKCYP2C19PREPFAPALDH1A1
SCHEMBL4051394 0.87 CTSK (0.34) CTSKPREPFAPELANEKMT2A
SCHEMBL4046884 0.87 CTSK (0.34) CTSKPREPFAPALDH1A1ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed