SCHEMBL4046064

SCHEMBL4046064

Cc1c(OC(=O)NC(Cc2cccs2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)c2ccc[n+]([O-])c2)oc2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 4/20 0.33
POLB P06746 1/20 0.32
CTSK P43235 3/20 0.32
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045719 0.91 SMN1; SMN2 (0.32) SMN1; SMN2CTSKCTSBCTSSCNR2
SCHEMBL4043622 0.90 CTSK (0.39) ALDH1A1CTSKCA12CA1CA2
SCHEMBL4040779 0.90 CTSV (0.34) SMN1; SMN2ALDH1A1CTSKUSP2GAA
SCHEMBL4050728 0.89 SMN1; SMN2 (0.33) SMN1; SMN2POLBCTSKUSP2GAA
SCHEMBL4045411 0.89 PREP (0.33) SMN1; SMN2ALDH1A1CTSKUSP2GAA
SCHEMBL4047038 0.87 CTSK (0.39) CTSKCTSBCTSS
SCHEMBL4046790 0.84 USP30 (0.36) CTSKCTSBCTSS
SCHEMBL4045248 0.84 NPC1 (0.33) SMN1; SMN2CTSKGAALMNAMAPT
SCHEMBL4046215 0.83 CHRNB2 (0.34) SMN1; SMN2CTSKUSP2GAALMNA
SCHEMBL4042344 0.83 CTSK (0.33) SMN1; SMN2ALDH1A1CTSKGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed