Water

Water

SCHEMBL4058718

O.O.O.O=C(O)CCN(CCN(CCC(=O)O)CC(=O)O)CC(=O)O

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.70
ADRA2A known ✓ P08913 1/20 0.70
SLC6A2 known ✓ P23975 1/20 0.70
SLC6A4 known ✓ P31645 1/20 0.70
ADRA1A known ✓ P35348 1/20 0.70
DRD3 known ✓ P35462 1/20 0.70
SLC6A3 known ✓ Q01959 1/20 0.70
ACE known ✓ P12821 1/20 0.65
LMNA P02545 3/20 0.70
TDP1 Q9NUW8 2/20 0.70
BLM P54132 2/20 0.70
PMP22 Q01453 2/20 0.70
KDM4E B2RXH2 1/20 0.70
ALOX15 P16050 1/20 0.70
TSHR P16473 1/20 0.70
DRD1 P21728 1/20 0.70
CYP2C19 P33261 1/20 0.70
HRH3 Q9Y5N1 1/20 0.70
EYA2 O00167 1/20 0.65
APP P05067 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10338095 0.97 LMNA (0.74) LMNATDP1BLMPMP22KDM4E
SCHEMBL2805867 0.97 LMNA (0.74) LMNATDP1BLMPMP22KDM4E
SCHEMBL13198811 0.95 TDP1 (0.79) LMNATDP1BLMPMP22KDM4E
SCHEMBL8663727 0.95 TDP1 (0.79) LMNATDP1BLMPMP22KDM4E
SCHEMBL29223102 0.95 LMNA (0.70) LMNATDP1BLMPMP22KDM4E
SCHEMBL562831 0.95 LMNA (0.68) LMNATDP1BLMPMP22KDM4E
SCHEMBL14315915 0.90 TDP1 (0.74) LMNATDP1BLMPMP22KDM4E
SCHEMBL21412890 0.90 TDP1 (0.74) LMNATDP1BLMPMP22KDM4E
Nitrilotriacetic Acid SCHEMBL9066282 0.90 TDP1 (0.65) LMNATDP1BLMPMP22KDM4E
SCHEMBL11636902 0.90 TDP1 (0.74) LMNATDP1BLMPMP22KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7524989-B2 Stabilized hydroxylamine solutions BASF AKTIENGESELLSCHAFT (DE) 2009-04-28 US claimed
EP-1434735-B1 STABILIZED HYDROXYLAMINE SOLUTIONS BASF AG (DE) 2006-10-25 EP claimed
US-20040242931-A1 Stabilized hydroxylamine solutions BASF AKTIENGESELLSCHAFT (DE) 2004-12-02 US claimed
US-5683793-A Ink jet transparencies XEROX CORPORATION (US) 1997-11-04 US claimed
US-7629400-B2 Image making medium HYMAN SYDNEY 2009-12-08 US disclosed
US-7524989-B2 Stabilized hydroxylamine solutions BASF AKTIENGESELLSCHAFT (DE) 2009-04-28 US disclosed
EP-1434735-B1 STABILIZED HYDROXYLAMINE SOLUTIONS BASF AG (DE) 2006-10-25 EP disclosed
US-20040242931-A1 Stabilized hydroxylamine solutions BASF AKTIENGESELLSCHAFT (DE) 2004-12-02 US disclosed
US-20030035917-A1 Image making medium HYMAN SYDNEY (US) 2003-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040242931-A1 Stabilized hydroxylamine solutions HNMT, HTT, BHMT CHRM2 1126/4885ADRA2A 95/4885SLC6A2 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.